SCHEMBL25990902

SCHEMBL25990902

O=Cc1ccc2noc(-c3cccc(C(F)(F)F)c3)c2c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.67
KDM4E B2RXH2 5/20 0.67
MEN1 O00255 3/20 0.67
KMT2A Q03164 3/20 0.67
POLB P06746 3/20 0.67
NPC1 O15118 2/20 0.67
IP6K1 Q92551 13/20 0.65
IP6K2 Q9UHH9 12/20 0.65
IP6K3 Q96PC2 11/20 0.65
SMN1; SMN2 Q16637 3/20 0.57
MAPT P10636 2/20 0.57
HPGD P15428 2/20 0.57
RAB9A P51151 1/20 0.57
PTK2B Q14289 1/20 0.57
HTT P42858 2/20 0.48
LMNA P02545 1/20 0.48
GAA P10253 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
TP53 P04637 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4934034 0.81 ALDH1A1 (1.00) ALDH1A1KDM4EMEN1KMT2APOLB
SCHEMBL25352733 0.81 KDM4E (0.73) ALDH1A1KDM4EMEN1KMT2APOLB
SCHEMBL6012040 0.81 ALDH1A1 (0.73) ALDH1A1KDM4EMEN1KMT2APOLB
SCHEMBL31265142 0.81 KDM4E (0.73) ALDH1A1KDM4EMEN1KMT2APOLB
SCHEMBL25990585 0.79 IP6K1 (1.00) ALDH1A1KDM4EMEN1KMT2APOLB
SCHEMBL30967420 0.79 IP6K1 (1.00) ALDH1A1KDM4EMEN1KMT2APOLB
SCHEMBL1814046 0.74 S1PR1 (0.68) IP6K1IP6K2IP6K3MAPT
SCHEMBL6199027 0.73 KDM4E (1.00) ALDH1A1KDM4EMEN1KMT2APOLB
SCHEMBL25353212 0.72 IP6K1 (0.80) ALDH1A1KDM4EMEN1KMT2APOLB
SCHEMBL7444196 0.72 CTSS (0.46) ALDH1A1KDM4EMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023154466-A1 ARYLBENZOISOXAZOLE COMPOUNDS AS IP6K AND IPMK INHIBITORS AND METHODS OF USE THEREOF THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2023-08-17 WO disclosed