SCHEMBL2600697

SCHEMBL2600697

C[C@@H](Cc1ccccc1)[C@H](O)CCl

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 3/20 0.69
CYP2D6 P10635 1/20 0.53
TAAR1 Q96RJ0 4/20 0.47
SIGMAR1 Q99720 4/20 0.47
SLC6A2 P23975 3/20 0.47
SLC6A4 P31645 2/20 0.47
SLC6A3 Q01959 2/20 0.47
MAOA P21397 1/20 0.47
CYP2A6 P11509 1/20 0.47
ADORA2A P29274 1/20 0.47
ADORA1 P30542 1/20 0.47
SLC18A2 Q05940 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
CYP1A2 P05177 1/20 0.41
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
HTR2A P28223 1/20 0.40
ADRA1A P35348 1/20 0.40
OPRK1 P41145 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14865966 1.00 TRPA1 (0.69) TRPA1CYP2D6TAAR1SIGMAR1SLC6A2
SCHEMBL8528186 0.84 TRPA1 (0.58) TRPA1CYP2D6TAAR1SIGMAR1SLC6A2
SCHEMBL16169480 0.82 TRPA1 (0.71) TRPA1CYP2D6TAAR1SIGMAR1SLC6A2
SCHEMBL18456337 0.82 TRPA1 (1.00) TRPA1CYP2D6TAAR1SIGMAR1SLC6A2
SCHEMBL12768230 0.82 TRPA1 (1.00) TRPA1CYP2D6TAAR1SIGMAR1SLC6A2
SCHEMBL14222474 0.81 TRPA1 (0.63) TRPA1CYP2D6TAAR1SIGMAR1SLC6A2
SCHEMBL19725385 0.81 TRPA1 (0.69) TRPA1CYP2D6TAAR1SIGMAR1SLC6A2
SCHEMBL21852752 0.81 TRPA1 (0.69) TRPA1CYP2D6TAAR1SIGMAR1SLC6A2
SCHEMBL234669 0.81 TRPA1 (0.69) TRPA1CYP2D6TAAR1SIGMAR1SLC6A2
SCHEMBL8263754 0.80 TRPA1 (0.69) TRPA1CYP2D6TAAR1SIGMAR1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9593073-B2 Method for the preparation of diazoalkanes BAKHU LIMITED (GB) 2017-03-14 US disclosed
US-20150038687-A1 METHOD FOR THE PREPARATION OF DIAZOALKANES BAKHU LIMITED (GB) 2015-02-05 US disclosed
US-20130116457-A1 CLEAN, HIGH-YIELD PREPARATION OF S,S AND R,S AMINO ACID ISOSTERES AEROJET FINE CHEMICALS LLC (US) 2013-05-09 US disclosed
US-20130096317-A1 REDUCTION OF ALDEHYDES AND KETONES TO ALCOHOLS GEORGIA TECH RESEARCH CORPORATION (US) 2013-04-18 US disclosed
US-8163933-B2 Clean, high-yield preparation of S,S and R,S amino acid isosteres AMPAC FINE CHEMICALS LLC (US) 2012-04-24 US disclosed
US-20090012303-A1 CLEAN, HIGH-YIELD PREPARATION OF S,S AND R,S AMINO ACID ISOSTERES AEROJET FINE CHEMICALS LLC (US) 2009-01-08 US disclosed
US-7309803-B2 Clean, High-yield preparation of S,S and R,S amino acid isosteres AEROJET FINE CHEMICALS LLC (US) 2007-12-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090012303-A1 CLEAN, HIGH-YIELD PREPARATION OF S,S AND R,S AMINO ACID ISOSTERES SRMS, HCK, BHMT2 TRPA1 4425/4885CYP2D6 1814/4885TAAR1 2357/4885
US-20150038687-A1 METHOD FOR THE PREPARATION OF DIAZOALKANES NIT2, DNTT, NAT1 TRPA1 1380/4885CYP2D6 185/4885TAAR1 324/4885
US-20130096317-A1 REDUCTION OF ALDEHYDES AND KETONES TO ALCOHOLS POF1B, PHF2, ADH1C TRPA1 3026/4885CYP2D6 1921/4885TAAR1 334/4885
US-20130116457-A1 CLEAN, HIGH-YIELD PREPARATION OF S,S AND R,S AMINO ACID ISOSTERES SRMS, HCK, BHMT2 TRPA1 4425/4885CYP2D6 1814/4885TAAR1 2357/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.