SCHEMBL26053296

SCHEMBL26053296

C#Cc1ccc2ccn(CCCC)c2c1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 2/20 0.57
CDK4 P11802 4/20 0.41
CCND1 P24385 4/20 0.41
CDC7 O00311 1/20 0.40
CDK2 P24941 1/20 0.40
MCL1 Q07820 4/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36
MTNR1A P48039 2/20 0.36
MTNR1B P49286 2/20 0.36
HTR1D P28221 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8430655 0.85 ALDH1A1 (0.46) HTR7CDK4CCND1CDC7CDK2
SCHEMBL24216449 0.84 HTR7 (0.56) HTR7CDC7CDK2HTR2AHTR2C
SCHEMBL8434667 0.76 HTR2C (0.56) HTR7CDK4CCND1HTR2AHTR2C
SCHEMBL27812843 0.76 CDK4 (0.44) CDK4CCND1MCL1HTR2AHTR2C
SCHEMBL8430623 0.76 KMO (0.59) HTR7CDK4CCND1MCL1HTR2A
SCHEMBL4651648 0.76 KDM4E (0.53) CDK4CCND1MCL1HTR2AHTR2C
SCHEMBL19526836 0.76 HTR7 (0.57) HTR7CDK4CCND1MCL1HTR2A
SCHEMBL18029368 0.75 HTR7 (0.49) HTR7CDC7CDK2
SCHEMBL8430662 0.75 ALDH1A1 (0.48) HTR7CDC7CDK2HTR2AHTR2C
SCHEMBL25154223 0.74 HTR7 (0.56) HTR7CDK4CCND1HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3931188-B1 NEW ISOINDOLINONE SUBSTITUTED INDOLES AND DERIVATIVES AS RAS INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2023-08-30 EP disclosed