SCHEMBL260737

SCHEMBL260737

Nc1nc2ccoc2c(=O)n1C1O[C@H](CO)[C@@H](O)[C@H]1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNP P00491 2/20 0.49
HSPA5 P11021 1/20 0.48
HSPA8 P11142 1/20 0.48
LMNA P02545 4/20 0.48
MTOR P42345 2/20 0.48
THRB P10828 1/20 0.48
MDM2 Q00987 1/20 0.48
NCOA1 Q15788 1/20 0.48
NCOA3 Q9Y6Q9 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.46
ALDH1A1 P00352 2/20 0.46
TP53 P04637 2/20 0.46
HBB P68871 2/20 0.46
POLB P06746 1/20 0.46
GMNN O75496 1/20 0.46
NFKB1 P19838 1/20 0.46
DNMT1 P26358 1/20 0.46
THPO P40225 1/20 0.46
HTT P42858 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL260036 0.78 ADORA2A (0.41) PNPLMNAMTORTHRBMDM2
SCHEMBL11291023 0.74 PNP (0.51) PNPHSPA5HSPA8LMNAMTOR
SCHEMBL12812951 0.72 LMNA (0.60) PNPHSPA5HSPA8LMNAMTOR
SCHEMBL12812953 0.72 LMNA (0.60) PNPHSPA5HSPA8LMNAMTOR
SCHEMBL7948397 0.71 PNP (0.54) PNPHSPA5HSPA8LMNAMTOR
SCHEMBL132926 0.71 PNP (0.54) PNPHSPA5HSPA8LMNAMTOR
SCHEMBL10496369 0.71 PNP (0.51) PNPHSPA5HSPA8LMNAMTOR
SCHEMBL10814776 0.71 PNP (0.54) PNPHSPA5HSPA8LMNAMTOR
SCHEMBL132927 0.71 PNP (0.51) PNPHSPA5HSPA8LMNAMTOR
SCHEMBL10496354 0.71 PNP (0.54) PNPHSPA5HSPA8LMNAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8133870-B2 Therapeutic furopyrimidines and thienopyrimidines BIOCRYST PHARMACEUTICALS, INC. (US) 2012-03-13 US claimed
US-20080300200-A1 Therapeutic Furopyrimidines and Thienopyrimidines BIOCRYST PHARMACEUTICALS, INC. (US) 2008-12-04 US claimed
US-20130078218-A1 HEPATITIS C THERAPIES BIOCRYST PHARMACEUTICALS, INC. 2013-03-28 US disclosed
EP-2537520-A1 Hepatics C therapies Biocryst Pharmaceuticals, Inc. (US) 2012-12-26 EP disclosed
US-20120213735-A1 THERAPEUTIC FUROPYRIMIDINES AND THIENOPYRIMIDINES BIOCRYST PHARMACEUTICALS, INC. (US) 2012-08-23 US disclosed
US-8163703-B2 Hepatitis C therapies BIOCRYST PHARMACEUTICALS, INC. (US) 2012-04-24 US disclosed
US-8133870-B2 Therapeutic furopyrimidines and thienopyrimidines BIOCRYST PHARMACEUTICALS, INC. (US) 2012-03-13 US disclosed
US-20100143300-A1 HEPATITIS C THERAPIES WILMINGTON TRUST, NATIONAL ASSOCIATION 2010-06-10 US disclosed
US-7514410-B2 Hepatitis C therapies BIOCRYST PHARMACEUTICALS, INC. (US) 2009-04-07 US disclosed
US-20080300200-A1 Therapeutic Furopyrimidines and Thienopyrimidines BIOCRYST PHARMACEUTICALS, INC. (US) 2008-12-04 US disclosed
US-20060234963-A1 Hepatitis C therapies WILMINGTON TRUST, NATIONAL ASSOCIATION 2006-10-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080300200-A1 Therapeutic Furopyrimidines and Thienopyrimidines DPYD, TYMP, TYMS PNP 23/4885HSPA5 2725/4885HSPA8 3461/4885
US-20130078218-A1 HEPATITIS C THERAPIES HAVCR2, FABP1, LIPC PNP 446/4885HSPA5 520/4885HSPA8 972/4885
US-20060234963-A1 Hepatitis C therapies HAVCR2, FABP1, LIPC PNP 446/4885HSPA5 520/4885HSPA8 972/4885
US-20120213735-A1 THERAPEUTIC FUROPYRIMIDINES AND THIENOPYRIMIDINES DPYD, TYMP, TYMS PNP 23/4885HSPA5 2725/4885HSPA8 3461/4885
US-20100143300-A1 HEPATITIS C THERAPIES HAVCR2, FABP1, LIPC PNP 446/4885HSPA5 520/4885HSPA8 972/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.