SCHEMBL26077458

SCHEMBL26077458

Cc1nc(-c2cc(Cl)cc(Cl)c2)cc(CO)c1F

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPV3 Q8NET8 1/20 0.38
NR4A2 P43354 1/20 0.34
MAPK1 P28482 1/20 0.32
MAP2K4 P45985 1/20 0.32
MAPKAPK2 P49137 1/20 0.32
MAPKAPK3 Q16644 1/20 0.32
MAPK6 Q16659 1/20 0.32
GCGR P47871 1/20 0.31
KMO O15229 1/20 0.30
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30931815 0.84 TRPV3 (0.36) TRPV3NR4A2KMO
SCHEMBL21550921 0.84 TRPV3 (0.36) TRPV3NR4A2KMO
SCHEMBL26077454 0.84 TRPV3 (0.34) TRPV3KMO
SCHEMBL21553800 0.83 TRPV3 (0.36) TRPV3NR4A2KMO
SCHEMBL30931827 0.83 TRPV3 (0.36) TRPV3NR4A2KMO
SCHEMBL26077459 0.76 SCN9A (0.33)
SCHEMBL21553744 0.71 SQOR (0.45)
SCHEMBL30931852 0.71 SQOR (0.45)
SCHEMBL26077457 0.71 SMN1; SMN2 (0.50)
SCHEMBL26077235 0.69 TRPV3 (0.35) TRPV3KMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11773078-B2 Furin inhibitors GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2023-10-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11773078-B2 Furin inhibitors FURIN, TGFB1, PCSK7 TRPV3 4541/4885NR4A2 3386/4885MAPK1 745/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.