SCHEMBL26085538

SCHEMBL26085538

C/N=C(\N)NC1CCOCC1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.38
NOS1 P29475 1/20 0.36
KDM1A O60341 1/20 0.31
NPSR1 Q6W5P4 3/20 0.31
MAPK1 P28482 2/20 0.31
CHEK1 O14757 1/20 0.31
CTSD P07339 2/20 0.31
CHRM4 P08173 1/20 0.30
MAPT P10636 2/20 0.30
ALDH1A1 P00352 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MCOLN3 Q8TDD5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20111343 0.80
SCHEMBL9060289 0.80 SIGMAR1 (0.58) SIGMAR1NOS1NPSR1MAPK1MAPT
SCHEMBL11301865 0.78 SIGMAR1 (0.61) SIGMAR1NPSR1MAPK1MAPTALDH1A1
SCHEMBL18619965 0.72 SIGMAR1 (0.36) SIGMAR1NOS1KDM4E
SCHEMBL4104793 0.71 KDM1A (0.33) KDM1ANPSR1MAPK1CHEK1MAPT
SCHEMBL16108920 0.71 ALDH1A1 (0.40) KDM1ANPSR1MAPK1CHEK1MAPT
SCHEMBL3644508 0.71 CHEK1 (0.41) KDM1ACHEK1CHRM4MAPTALDH1A1
SCHEMBL29131058 0.70 POLB (0.57) MAPK1ALDH1A1
Hydrochloric Acid SCHEMBL18281392 0.70 KDM1A (0.33) KDM1ANPSR1MAPK1CHEK1MAPT
SCHEMBL3141240 0.68 NPC1 (0.43) KDM1AMAPK1CHEK1CHRM4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3307727-B1 HETEROCYCLIC INHIBITORS OF ERK1 AND ERK2 AND THEIR USE IN THE TREATMENT OF CANCER ASANA BIOSCIENCES LLC (US) 2023-10-04 EP disclosed