SCHEMBL26088656

SCHEMBL26088656

NC(=S)N/N=C\CC1COC1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
KDM4E B2RXH2 1/20 0.35
MAOA P21397 1/20 0.35
RAB9A P51151 1/20 0.32
GAA P10253 1/20 0.32
POLB P06746 1/20 0.32
CTSK P43235 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26091858 1.00 ALDH1A1 (0.46) ALDH1A1NPSR1KDM4EMAOARAB9A
SCHEMBL7338693 0.72 ALDH1A1 (0.44) ALDH1A1NPSR1KDM4EMAOAGAA
SCHEMBL26090195 0.72 KDM4E (0.38) ALDH1A1NPSR1KDM4EMAOARAB9A
SCHEMBL7910374 0.66
SCHEMBL7910372 0.66
SCHEMBL20821435 0.64
SCHEMBL17666902 0.63
SCHEMBL17666901 0.63
SCHEMBL11672130 0.62 MAOA (0.42) ALDH1A1NPSR1KDM4EMAOA
SCHEMBL1642699 0.61 KDM4E (0.52) NPSR1KDM4EGAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023067515-A1 THIADIAZOLYL COMPOUNDS AS DNA POLYMERASE THETA INHIBITORS IDEAYA BIOSCIENCES, INC. (US) 2023-04-27 WO disclosed
WO-2023067515-A1 THIADIAZOLYL COMPOUNDS AS DNA POLYMERASE THETA INHIBITORS IDEAYA BIOSCIENCES, INC. (US) 2023-04-27 WO disclosed