SCHEMBL26089403

SCHEMBL26089403

O=C(Cc1ccc2c(c1)OCO2)Nc1ccc2c(c1)S(=O)(=O)C=C2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.52
CA12 O43570 1/20 0.50
CA9 Q16790 1/20 0.50
ALDH1A1 P00352 5/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
HTT P42858 1/20 0.48
MAPT P10636 2/20 0.47
MAPK8 P45983 1/20 0.47
NPC1 O15118 1/20 0.46
STAT3 P40763 1/20 0.46
LMNA P02545 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
KDM4E B2RXH2 1/20 0.46
KMT2A Q03164 1/20 0.45
GAA P10253 1/20 0.45
EPHX2 P34913 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30346013 0.94 MAPT (0.52) RAB9ACA12CA9ALDH1A1SMN1; SMN2
SCHEMBL26087395 0.94 MAPT (0.52) RAB9ACA12CA9ALDH1A1SMN1; SMN2
SCHEMBL26089410 0.89 RAB9A (0.52) RAB9ACA12CA9ALDH1A1SMN1; SMN2
SCHEMBL26090717 0.84 CA12 (0.45) RAB9ACA12CA9ALDH1A1SMN1; SMN2
SCHEMBL26087397 0.83 GAA (0.52) RAB9ACA12CA9ALDH1A1SMN1; SMN2
SCHEMBL179015 0.82 RAB9A (0.71) RAB9AALDH1A1SMN1; SMN2HTTMAPT
SCHEMBL30346080 0.80 MEN1 (0.53) ALDH1A1SMN1; SMN2HTTMAPTSTAT3
SCHEMBL30346152 0.80 STAT3 (0.48) RAB9ACA12CA9ALDH1A1SMN1; SMN2
SCHEMBL30345669 0.80 ALDH1A1 (0.52) CA12CA9ALDH1A1SMN1; SMN2HTT
SCHEMBL26087977 0.80 STAT3 (0.48) RAB9ACA12CA9ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023068852-A1 BENZOTHIOPHENE-1,1-DIOXIDE DERIVATIVE COMPOUND AS STAT3 INHIBITOR, AND USE THEREOF 주식회사 프롬바이오 2023-04-27 WO claimed
WO-2023068852-A1 BENZOTHIOPHENE-1,1-DIOXIDE DERIVATIVE COMPOUND AS STAT3 INHIBITOR, AND USE THEREOF 주식회사 프롬바이오 2023-04-27 WO disclosed