SCHEMBL26102005

SCHEMBL26102005

CC(C)(C)C1(c2cc(C#N)ccc2C(=O)N2CCC(OC(F)(F)F)CC2)C=CN=N1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 2/20 0.41
CACNA1B Q00975 2/20 0.41
SMO Q99835 2/20 0.38
HCRTR1 O43613 3/20 0.36
HCRTR2 O43614 3/20 0.36
KDM1A O60341 1/20 0.36
FASN P49327 7/20 0.36
GPR119 Q8TDV5 2/20 0.34
RBP4 P02753 1/20 0.34
RORC P51449 1/20 0.34
SLC6A9 P48067 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26099432 0.87 NR1I2 (0.41) NR1I2CACNA1BSMOFASNRORC
SCHEMBL26101807 0.81 NR1I2 (0.36) NR1I2CACNA1BHCRTR1HCRTR2FASN
SCHEMBL26099356 0.76 NR1I2 (0.42) NR1I2CACNA1BSMOHCRTR1HCRTR2
SCHEMBL30429790 0.76 NR1I2 (0.42) NR1I2CACNA1BSMOHCRTR1HCRTR2
SCHEMBL26104159 0.76 SLC22A12 (0.35)
SCHEMBL30430028 0.75 MBTD1 (0.42) NR1I2CACNA1BSMOHCRTR1HCRTR2
SCHEMBL26102446 0.75 CFTR (0.34) HCRTR1HCRTR2
SCHEMBL26100540 0.75 MBTD1 (0.42) NR1I2CACNA1BSMOHCRTR1HCRTR2
SCHEMBL26105235 0.74 NR1I2 (0.39) NR1I2CACNA1BSMOFASNRBP4
SCHEMBL26102345 0.74 FASN (0.38) NR1I2CACNA1BSMOHCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023076219-A2 ANTAGONISTS OF GPR39 PROTEIN VASOCARDEA, INC. (US) 2023-05-04 WO disclosed