SCHEMBL26099356

SCHEMBL26099356

N#Cc1ccc(C(=O)N2CCC(OC(F)(F)F)CC2)c(B(O)O)c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 2/20 0.42
CACNA1B Q00975 2/20 0.42
SMO Q99835 1/20 0.41
PDK1 Q15118 1/20 0.41
PDK2 Q15119 1/20 0.41
PDK3 Q15120 1/20 0.41
PDK4 Q16654 1/20 0.41
POLB P06746 1/20 0.41
KDM1A O60341 3/20 0.40
FASN P49327 4/20 0.40
GPR119 Q8TDV5 1/20 0.39
SLC6A9 P48067 6/20 0.39
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
KCNH2 Q12809 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30429790 1.00 NR1I2 (0.42) NR1I2CACNA1BSMOPDK1PDK2
SCHEMBL30430028 0.85 MBTD1 (0.42) NR1I2CACNA1BSMOPOLBKDM1A
SCHEMBL26100540 0.85 MBTD1 (0.42) NR1I2CACNA1BSMOPOLBKDM1A
SCHEMBL30430006 0.78 NR1I2 (0.39) NR1I2CACNA1BSMOKDM1AFASN
SCHEMBL26104208 0.76 SLC6A9 (0.41) PDK1PDK2PDK3PDK4FASN
SCHEMBL30430083 0.76 SLC6A9 (0.41) PDK1PDK2PDK3PDK4FASN
SCHEMBL26102005 0.76 NR1I2 (0.41) NR1I2CACNA1BSMOKDM1AFASN
SCHEMBL30430098 0.75 HSD11B1 (0.59) SMOPOLBHCRTR1HCRTR2
SCHEMBL26103330 0.72 RORC (0.47) POLBKDM1AFASNGPR119
SCHEMBL30396527 0.71 SCD (0.44) NR1I2CACNA1BSMOFASNSLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023076219-A2 ANTAGONISTS OF GPR39 PROTEIN VASOCARDEA, INC. (US) 2023-05-04 WO disclosed
WO-2023076219-A2 ANTAGONISTS OF GPR39 PROTEIN VASOCARDEA, INC. (US) 2023-05-04 WO disclosed