SCHEMBL261676

SCHEMBL261676

C1=C2C(=Nc3ccccc32)c2ccccc21

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.62
IDO1 P14902 1/20 0.41
MAPT P10636 3/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
APAF1 O14727 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
TSHR P16473 1/20 0.36
HK1 P19367 1/20 0.36
GALK1 P51570 1/20 0.36
HKDC1 Q2TB90 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SRC P12931 2/20 0.33
CTRB1 P17538 2/20 0.33
CCNE1 P24864 2/20 0.33
CDK2 P24941 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30019213 1.00 ABCG2 (0.62) ABCG2IDO1MAPTALDH1A1MEN1
SCHEMBL7464999 0.85 ABCG2 (0.55) ABCG2IDO1MAPTALDH1A1MEN1
SCHEMBL4499072 0.83 ABCG2 (0.46) ABCG2IDO1MAPTALDH1A1MEN1
SCHEMBL4510312 0.82 ABCG2 (0.45) ABCG2IDO1MAPTALDH1A1MEN1
SCHEMBL7733305 0.80 ABCG2 (0.50) ABCG2ALDH1A1TSHRHSD17B10MAPK1
SCHEMBL1820361 0.77 ABCG2 (0.68) ABCG2IDO1MAPTALDH1A1MEN1
SCHEMBL4313626 0.77 ABCG2 (0.68) ABCG2IDO1MAPTALDH1A1MEN1
SCHEMBL725971 0.77 ABCG2 (0.51) ABCG2IDO1
SCHEMBL1899423 0.77 ABCG2 (0.68) ABCG2IDO1MAPTALDH1A1MEN1
SCHEMBL527160 0.76 ABCG2 (0.46) ABCG2IDO1MAPTALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 108 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108503578-A A kind of synthetic method of indeno-[1,2-b] indoles -10 (5H) -one class compound 中国烟草总公司郑州烟草研究院 2018-09-07 CN claimed
US-20240392044-A1 OLEFIN POLYMERIZATION CATALYST SYSTEM AND POLYMERIZATION PROCESS NOVA CHEMICALS (INTERNATIONAL) S.A. (CH) 2024-11-28 US disclosed
EP-4405367-A1 OLEFIN POLYMERIZATION CATALYST SYSTEM AND POLYMERIZATION PROCESS Nova Chemicals (International) S.A. (CH) 2024-07-31 EP disclosed
WO-2023042155-A1 OLEFIN POLYMERIZATION CATALYST SYSTEM AND POLYMERIZATION PROCESS NOVA CHEMICALS (INTERNATIONAL) S.A. (CH) 2023-03-23 WO disclosed
CN-108503578-A A kind of synthetic method of indeno-[1,2-b] indoles -10 (5H) -one class compound 中国烟草总公司郑州烟草研究院 2018-09-07 CN disclosed
CN-108503578-A A kind of synthetic method of indeno-[1,2-b] indoles -10 (5H) -one class compound 中国烟草总公司郑州烟草研究院 2018-09-07 CN disclosed
JP-5371763-B2 2013-12-18 JP disclosed
EP-2079691-B1 SUBSTITUTED INDENO[1,2-B]INDOLE DERIVATIVES AS NOVEL INHIBITORS OF PROTEIN KINASE CK2 AND THEIR USE AS TUMOUR THERAPEUTIC AGENTS, CYTOSTATICS AND DIAGNOSTIC AIDS UNIV DUESSELDORF H HEINE (DE) 2013-08-14 EP disclosed
US-8252814-B2 Agents and crystals for improving excretory potency of urinary bladder TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-08-28 US disclosed
US-8133913-B2 Substituted indeno [1,2-b]indole derivatives as novel inhibitors of protein kinase CK2 and their use as tumor therapeutic agents, cytostatics and diagnostic aids Heinrich-Heine Universitat Dusseldof (DE) 2012-03-13 US disclosed
US-6391902-B2 TREATMENT OF DISORDERS ASSOCIATED WITH SMOOTH MUSCLE CONTRACTION SUCH AS INCONTINENCE AND IRRITABLE BOWEL SYNDROME AMERICAN HOME PRODUCTS CORPORATION 2002-05-21 US disclosed
US-6376629-B2 ORGANOMETALLIC COMPOUND EQUISTAR CHEMICALS, LP 2002-04-23 US disclosed
US-20010047026-A1 Substituted benzofuranoindoles and indenoindoles as novel potassium channel openers AMERICAN HOME PRODUCTS CORPORATION 2001-11-29 US disclosed
US-6288099-B1 COMPOUNDS SUCH AS 8-BROMO-10H-BENZO(4,5)FURO(3,2-B)INDOLE-1-CARBOXYLIC ACID USED TO TREAT DISORDERS ASSOCIATED WITH SMOOTH MUSCLE CONTRATION SUCH AS URINARY INCONTINENCE AND IRRITABLE BOWL SYNDROME AMERICAN HOME PRODUCTS CORPORATION 2001-09-11 US disclosed
EP-1118322-A1 DRUGS FOR IMPROVING VESICAL EXCRETORY STRENGTH Takeda Chemical Industries, Ltd. (JP) 2001-07-25 EP disclosed
US-20010007848-A1 Single-site catalysts for olefin polymerization EQUISTAR CHEMICALS, L.P. 2001-07-12 US disclosed
US-6232260-B1 ORGANOMETALLIC COMPLEX COMPRISES A GROUP 3 TO 10 TRANSITION OR LANTHANIDE METAL, M, AND AT LEAST ONE INDENOINDOLYL LIGAND THAT IS .PI.-BONDED TO M. EQUISTAR CHEMICALS, L.P. 2001-05-15 US disclosed
WO-2001027125-A1 SINGLE-SITE CATALYSTS FOR OLEFIN POLYMERIZATION EQUISTAR CHEMICALS, L.P. (US) 2001-04-19 WO disclosed
US-5620973-A CHOLINESTERASE INHIBITOR; ALZHEIMER*S DISEASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-15 US disclosed
EP-0655451-A1 Tetracyclic condensed heterocyclic compounds for the treatment of senile dementia TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-05-31 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010047026-A1 Substituted benzofuranoindoles and indenoindoles as novel potassium channel openers KCNJ2, KCNN3, KCNN2 ABCG2 904/4885IDO1 1016/4885MAPT 4000/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.