SCHEMBL262073

SCHEMBL262073

COC(=O)[C@H](C)c1ccc(NC(N)=S)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
HPGD P15428 3/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
ALOX12 P18054 1/20 0.47
CYP2C19 P33261 1/20 0.47
KIF11 P52732 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
KMT2A Q03164 2/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
TP53 P04637 1/20 0.43
TYR P14679 1/20 0.43
TSHR P16473 1/20 0.43
TAS2R38 P59533 1/20 0.43
HSD17B10 Q99714 1/20 0.43
MEN1 O00255 1/20 0.43
RAB9A P51151 1/20 0.43
GLA P06280 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2171946 1.00 ALDH1A1 (0.47) ALDH1A1HPGDCYP3A4CYP2D6CYP2C9
SCHEMBL2170844 1.00 ALDH1A1 (0.47) ALDH1A1HPGDCYP3A4CYP2D6CYP2C9
SCHEMBL2170717 0.87 KIF11 (0.60) ALDH1A1HPGDKIF11SMN1; SMN2KMT2A
SCHEMBL2172524 0.87 KIF11 (0.60) ALDH1A1HPGDKIF11SMN1; SMN2KMT2A
SCHEMBL261230 0.87 KIF11 (0.60) ALDH1A1HPGDKIF11SMN1; SMN2KMT2A
SCHEMBL2170471 0.83 NR1H4 (0.54) ALDH1A1HPGDCYP3A4CYP2D6CYP2C9
SCHEMBL2815572 0.83 NR1H4 (0.54) ALDH1A1HPGDCYP3A4CYP2D6CYP2C9
SCHEMBL1447652 0.81 SMN1; SMN2 (0.56) ALDH1A1HPGDCYP3A4CYP2C19SMN1; SMN2
SCHEMBL11272564 0.78 HPGD (0.49) ALDH1A1HPGDCYP3A4SMN1; SMN2KMT2A
SCHEMBL5523228 0.77 KIF11 (0.59) ALDH1A1HPGDCYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8133911-B2 (R)-4-(heteroaryl) phenylethyl derivatives and pharmaceutical compositions containing them DOMPE S.P.A (IT) 2012-03-13 US disclosed
EP-2201006-B1 (R)-4-(HETEROARYL) PHENYLETHYL DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DOMPE SPA (IT) 2011-03-09 EP disclosed