SCHEMBL26258443

SCHEMBL26258443

CCNC(=O)NC(C)Cc1ccccc1

nearest known ligand 0.77

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.77
RAB9A P51151 2/20 0.77
LMNA P02545 1/20 0.67
ACACB O00763 1/20 0.59
OPRM1 P35372 7/20 0.58
OPRK1 P41145 5/20 0.58
OPRD1 P41143 4/20 0.58
TAAR1 Q96RJ0 1/20 0.56
EPHX2 P34913 2/20 0.56
SIGMAR1 Q99720 1/20 0.56
GAA P10253 1/20 0.55
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12204095 1.00 NPC1 (0.77) NPC1RAB9ALMNAACACBOPRM1
SCHEMBL14654946 0.88 NPC1 (1.00) NPC1RAB9ALMNAOPRM1OPRK1
SCHEMBL10429991 0.83 LMNA (0.67) LMNAGAAKMT2A
SCHEMBL11581315 0.83 NPC1 (0.83) NPC1RAB9ALMNAOPRM1OPRK1
SCHEMBL7445998 0.81 CAPN1 (0.55) NPC1RAB9A
SCHEMBL24609344 0.80 NPC1 (0.79) NPC1RAB9ALMNATAAR1SIGMAR1
SCHEMBL2543698 0.80 NPC1 (0.79) NPC1RAB9ALMNATAAR1SIGMAR1
SCHEMBL21992681 0.80 NPC1 (0.67) NPC1RAB9ALMNAOPRM1OPRK1
SCHEMBL11580858 0.80 NPC1 (0.77) NPC1RAB9ALMNATAAR1EPHX2
SCHEMBL7445995 0.80 NPC1 (0.49) NPC1RAB9ALMNAACACBEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230285570-A1 THERAPEUTICALLY USEFUL CURE-PRO MOLECULES FOR E3 LIGASE MEDIATED DEGRADATION OF PROTEINS, AND METHODS OF MAKING AND USING THEM CORNELL UNIVERSITY 2023-09-14 US disclosed
US-20230277553-A1 THERAPEUTIC COMPOSITION OF CURE-PRO COMPOUNDS FOR TARGETED DEGRADATION OF BET DOMAIN PROTEINS, AND METHODS OF MAKING AND USAGE CORNELL UNIVERSITY 2023-09-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230285570-A1 THERAPEUTICALLY USEFUL CURE-PRO MOLECULES FOR E3 LIGASE MEDIATED DEGRADATION OF PROTEINS, AND METHODS OF MAKING AND USING THEM XIAP, CUL4A, CUL1 NPC1 3588/4885RAB9A 3063/4885LMNA 1674/4885
US-20230277553-A1 THERAPEUTIC COMPOSITION OF CURE-PRO COMPOUNDS FOR TARGETED DEGRADATION OF BET DOMAIN PROTEINS, AND METHODS OF MAKING AND USAGE BET1, BRD4, PHKB NPC1 3741/4885RAB9A 3432/4885LMNA 1366/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.