SCHEMBL263098

SCHEMBL263098

Cc1noc(C)c1C([O])=O

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
LMNA P02545 1/20 0.47
GAA P10253 2/20 0.45
ALOX15 P16050 3/20 0.44
GFER P55789 1/20 0.44
TSHR P16473 3/20 0.42
HSD17B10 Q99714 2/20 0.42
USP2 O75604 1/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
KDM4E B2RXH2 2/20 0.41
ATM Q13315 1/20 0.41
MAPT P10636 1/20 0.41
AGTR1 P30556 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL223413 0.81 GAA (0.49) ALDH1A1L3MBTL1LMNAGAAALOX15
SCHEMBL358889 0.81 ALDH1A1 (0.47) ALDH1A1L3MBTL1LMNAGAAALOX15
SCHEMBL193631 0.79 LMNA (0.50) ALDH1A1L3MBTL1LMNAGAAALOX15
SCHEMBL352276 0.79 GAA (0.53) ALDH1A1L3MBTL1LMNAGAAALOX15
SCHEMBL3643406 0.79 ALDH1A1 (0.46) ALDH1A1L3MBTL1LMNAGAAALOX15
Hydrochloric Acid SCHEMBL19119186 0.79 GAA (0.47) ALDH1A1L3MBTL1LMNAGAAALOX15
SCHEMBL2176508 0.77 ALDH1A1 (0.45) ALDH1A1L3MBTL1LMNAGAAALOX15
Hydrochloric Acid SCHEMBL5009791 0.77 GAA (0.51) ALDH1A1L3MBTL1LMNAGAAALOX15
SCHEMBL8571245 0.76 GFER (0.47) ALDH1A1L3MBTL1LMNAGAAALOX15
SCHEMBL14676577 0.76 HPGD (0.56) ALDH1A1L3MBTL1ALOX15TSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2254416-B1 HERBICIDAL COMPOUNDS SYNGENTA LTD (GB) 2016-09-07 EP disclosed
US-8987455-B2 Herbicidal compounds SYNGENTA LIMITED (GB) 2015-03-24 US disclosed
US-8653078-B2 Herbicidal pyrido[2,3-b]pyrazines SYNGENTA LIMITED 2014-02-18 US disclosed
US-8557840-B2 Herbicidal compounds SYNGENTA LIMITED (GB) 2013-10-15 US disclosed
US-20130137574-A1 HERBICIDAL COMPOUNDS SYNGENTA LIMITED (GB) 2013-05-30 US disclosed
US-8338598-B2 Herbicidal pyrido[2,3-B]pyrazines and their use as herbicides SYNGENTA LIMITED 2012-12-25 US disclosed
EP-2057154-B1 PYRIDO [2, 3-B]PYRAZINE DERIVATIVES USEFUL AS HERBICIDAL COMPOUNDS SYNGENTA LTD (GB) 2012-11-14 EP disclosed
US-8217055-B2 Pyrido-pyrazine derivatives useful as herbicidal compounds SYNGENTA CROP PROTECTION LLC (US) 2012-07-10 US disclosed
US-8133847-B2 Pyrido[2,3-B]pyrazine derivatives useful as herbicidal compounds SYNGENTA LIMITED (GB) 2012-03-13 US disclosed
US-20110034334-A1 HERBICIDAL COMPOUNDS SYNGENTA CROP PROTECTION, INC. (US) 2011-02-10 US disclosed
US-20110021351-A1 HERBICIDAL COMPOUNDS SYNGENTA CROP PROTECTION, INC. (US) 2011-01-27 US disclosed
EP-2254417-A2 HERBICIDAL COMPOUNDS Syngenta Limited (GB) 2010-12-01 EP disclosed
EP-2254416-A2 HERBICIDAL COMPOUNDS Syngenta Limited (GB) 2010-12-01 EP disclosed
EP-2102205-B1 PYRIDO-PYRAZINE DERIVATIVES USEFUL AS HERBICIDAL COMPOUNDS SYNGENTA LTD (GB) 2010-09-01 EP disclosed
US-20100167929-A1 PYRIDO-PYRAZINE DERIVATIVES USEFUL AS HERBICIDAL COMPOUNDS SYNGENTA CROP PROTECTION, INC. (US) 2010-07-01 US disclosed
US-20090305892-A1 PYRIDO[2,3-B]PYRAZINE DERIVATIVES USEFUL AS HERBICIDAL COMPOUNDS SYNGENTA LIMITED (GB) 2009-12-10 US disclosed
WO-2009090402-A2 HERBICIDAL COMPOUNDS SYNGENTA LIMITED (GB) 2009-07-23 WO disclosed
WO-2009090401-A2 HERBICIDAL COMPOUNDS SYNGENTA LIMITED (GB) 2009-07-23 WO disclosed
EP-2057154-A1 PYRIDO [2, 3-B]PYRAZINE DERIVATIVES USEFUL AS HERBICIDAL COMPOUNDS Syngenta Limited (GB) 2009-05-13 EP disclosed
WO-2008009908-A1 PYRIDO [2, 3-B] PYRAZINE DERIVATIVES USEFUL AS HERBICIDAL COMPOUNDS SYNGENTA LIMITED (GB) 2008-01-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130137574-A1 HERBICIDAL COMPOUNDS DDT, CBR3, CBR1 ALDH1A1 133/4885L3MBTL1 3016/4885LMNA 3807/4885
US-20100167929-A1 PYRIDO-PYRAZINE DERIVATIVES USEFUL AS HERBICIDAL COMPOUNDS CBR3, PNPO, CBR1 ALDH1A1 354/4885L3MBTL1 2960/4885LMNA 3893/4885
US-20110021351-A1 HERBICIDAL COMPOUNDS DDT, CBR3, TH ALDH1A1 299/4885L3MBTL1 3091/4885LMNA 3883/4885
US-20110034334-A1 HERBICIDAL COMPOUNDS CYP4Z1, CYP4F3, DDT ALDH1A1 119/4885L3MBTL1 2349/4885LMNA 2904/4885
US-20090305892-A1 PYRIDO[2,3-B]PYRAZINE DERIVATIVES USEFUL AS HERBICIDAL COMPOUNDS PNPO, CBR3, CBR1 ALDH1A1 286/4885L3MBTL1 1707/4885LMNA 3694/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.