SCHEMBL2636367

SCHEMBL2636367

COc1cccc([C@](C)(O)I)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.50
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
ENPP2 Q13822 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP3A4 P08684 1/20 0.44
KIF11 P52732 1/20 0.43
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
LMNA P02545 2/20 0.42
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42
STAT1 P42224 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PDK1 Q15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23343726 0.84 ACHE (0.48) ACHECES2CES1ENPP2CA1
SCHEMBL6897457 0.84 ACHE (0.48) ACHECES2CES1ENPP2CA1
SCHEMBL8367527 0.84 ACHE (0.48) ACHECES2CES1ENPP2CA1
SCHEMBL2534644 0.84 ACHE (0.48) ACHECES2CES1ENPP2CA1
SCHEMBL22932513 0.82 ACHE (0.50) ACHECES2CES1ENPP2CA1
SCHEMBL18535826 0.81 KIF11 (0.48) ACHECES2CES1ENPP2CA1
SCHEMBL3973199 0.81 KIF11 (0.50) ACHECES2CES1ENPP2CA1
SCHEMBL5324674 0.81 KIF11 (0.50) ACHECES2CES1ENPP2CA1
SCHEMBL4874637 0.81 KIF11 (0.50) ACHECES2CES1ENPP2CA1
SCHEMBL14919359 0.80 ACHE (0.48) ACHECES2CES1ENPP2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2438048-A2 POLYCYCLIC ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS Amira Pharmaceuticals, Inc. (US) 2012-04-11 EP disclosed
WO-2010141761-A2 POLYCYCLIC ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-12-09 WO disclosed