SCHEMBL14919359

SCHEMBL14919359

COc1cccc(C(C)(C)F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.48
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP3A4 P08684 1/20 0.47
NPSR1 Q6W5P4 2/20 0.45
MAPT P10636 2/20 0.45
KIF11 P52732 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
PDK1 Q15118 1/20 0.44
PDK2 Q15119 1/20 0.44
PDK3 Q15120 1/20 0.44
PDK4 Q16654 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL167016 0.85 L3MBTL1 (0.58) ACHECA1CA2CA7CA9
SCHEMBL29782607 0.85 L3MBTL1 (0.58) ACHECA1CA2CA7CA9
SCHEMBL27295380 0.83 MAPT (0.57) ACHECA1CA2CA7CA9
SCHEMBL8408204 0.83 ACHE (0.52) ACHECA1CA2CA7CA9
SCHEMBL146154 0.83 ACHE (0.52) ACHECA1CA2CA7CA9
SCHEMBL14920642 0.82 ALDH1A1 (0.50) ACHECA1CA2CA7CA9
SCHEMBL14191200 0.82 ACHE (0.47) ACHECA1CA2CA7CA9
SCHEMBL13019342 0.82 KIF11 (0.47) ACHECA1CA2CA7CA9
SCHEMBL23838094 0.81 HSD11B1 (0.50) ACHECA1CA2CA7CA9
SCHEMBL21087697 0.81 HSD11B1 (0.50) ACHECA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2773210-A1 PROCESS FOR A CETP INHIBITOR Merck Sharp & Dohme Corp. (US) 2014-09-10 EP disclosed
WO-2013066768-A1 PROCESS FOR A CETP INHIBITOR MERCK SHARP & DOHME CORP. (US) 2013-05-10 WO disclosed