SCHEMBL3973199

SCHEMBL3973199

COc1cccc([C@@](C)(N)I)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.50
ALDH1A1 P00352 1/20 0.48
CYP3A4 P08684 1/20 0.48
ACHE P22303 1/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
TAAR1 Q96RJ0 4/20 0.42
IDO1 P14902 2/20 0.42
AGXT P21549 2/20 0.42
PARP1 P09874 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PRSS1 P07477 1/20 0.42
PRSS2 P07478 1/20 0.42
PRSS3 P35030 1/20 0.42
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
HTR3A P46098 1/20 0.41
HTR3D Q70Z44 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4874637 1.00 KIF11 (0.50) KIF11ALDH1A1CYP3A4ACHECA1
SCHEMBL5324674 1.00 KIF11 (0.50) KIF11ALDH1A1CYP3A4ACHECA1
SCHEMBL23343726 0.84 ACHE (0.48) KIF11ALDH1A1CYP3A4ACHECA1
SCHEMBL2060637 0.84 ALDH1A1 (0.52) KIF11ALDH1A1CYP3A4ACHECA1
Hydrochloric Acid SCHEMBL30324798 0.82 ALDH1A1 (0.50) KIF11ALDH1A1CYP3A4ACHECA1
Hydrochloric Acid SCHEMBL29240545 0.82 ALDH1A1 (0.50) KIF11ALDH1A1CYP3A4ACHECA1
SCHEMBL2636367 0.81 ACHE (0.50) KIF11ALDH1A1CYP3A4ACHECA1
SCHEMBL7884887 0.81 ALDH1A1 (0.48) KIF11ALDH1A1CYP3A4ACHECA1
SCHEMBL8408204 0.79 ACHE (0.52) KIF11ALDH1A1CYP3A4ACHECA1
SCHEMBL146154 0.79 ACHE (0.52) KIF11ALDH1A1CYP3A4ACHECA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074120-A1 TROPANE COMPOUNDS Exelixis, Inc. (US) 2009-07-01 EP disclosed
WO-2009055077-A1 TROPANE COMPOUNDS EXELIXIS, INC. (US) 2009-04-30 WO disclosed
WO-2007109615-A2 β -LACTAMYL VASOPRESSIN V2 ANTAGONISTS AZEVAN PHARMACEUTICALS, INC. (US) 2007-09-27 WO disclosed