SCHEMBL2637445

SCHEMBL2637445

O=C(Nc1cc[nH]n1)c1c(=O)[nH]n2c(=O)cc(-c3ccccc3)[nH]c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
ERCC1 P07992 1/20 0.36
FEN1 P39748 1/20 0.36
ERCC4 Q92889 1/20 0.36
ALPL P05186 1/20 0.36
ALPI P09923 1/20 0.36
MAPT P10636 2/20 0.35
ALDH1A1 P00352 3/20 0.35
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
LMNA P02545 1/20 0.35
PKM P14618 1/20 0.35
MAPK1 P28482 1/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
DHODH Q02127 2/20 0.34
MAT2A P31153 2/20 0.34
POLB P06746 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2637450 0.89 MEN1 (0.38) NPC1RAB9AKMT2AMEN1MAPK1
SCHEMBL2637908 0.84 NPC1 (0.45) NPC1RAB9AMAPTALDH1A1KMT2A
SCHEMBL2638043 0.83 MAPK10 (0.45) NPC1RAB9AERCC1FEN1ERCC4
SCHEMBL2640983 0.83 ALDH1A1 (0.47) NPC1RAB9AERCC1FEN1ERCC4
SCHEMBL2637520 0.80 DHODH (0.45) NPC1RAB9AERCC1FEN1ERCC4
SCHEMBL2637918 0.79 KMT2A (0.41) NPC1RAB9AERCC1FEN1ERCC4
SCHEMBL2637500 0.78 ALDH1A1 (0.39) ERCC1FEN1ERCC4MAPTALDH1A1
SCHEMBL2637350 0.78 ERCC1 (0.48) NPC1RAB9AERCC1FEN1ERCC4
SCHEMBL2637610 0.78 MAPK8 (0.48) NPC1RAB9AMAPTALDH1A1KMT2A
SCHEMBL2637592 0.77 MEN1 (0.45) NPC1RAB9AALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2438070-A1 GLYCINE B ANTAGONISTS Merz Pharma GmbH & Co. KGaA (DE) 2012-04-11 EP claimed
WO-2010139483-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2010-12-09 WO claimed
EP-2438070-A1 GLYCINE B ANTAGONISTS Merz Pharma GmbH & Co. KGaA (DE) 2012-04-11 EP disclosed
WO-2010139483-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2010-12-09 WO disclosed