SCHEMBL2640983

SCHEMBL2640983

O=C(Nc1ccon1)c1c(=O)[nH]n2c(=O)cc(-c3ccccc3)[nH]c12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
KMT2A Q03164 3/20 0.43
HPGD P15428 3/20 0.43
KDM4E B2RXH2 2/20 0.43
TSHR P16473 2/20 0.43
MEN1 O00255 2/20 0.43
USP2 O75604 1/20 0.43
MAPK1 P28482 1/20 0.43
HSD17B10 Q99714 1/20 0.43
SMN1; SMN2 Q16637 6/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GAA P10253 1/20 0.40
TP53 P04637 1/20 0.40
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
LMNA P02545 1/20 0.37
ALPL P05186 2/20 0.37
ALPI P09923 2/20 0.37
ALPG P10696 2/20 0.37
ERCC1 P07992 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2637249 0.89 SMN1; SMN2 (0.50) ALDH1A1KMT2AHPGDKDM4ETSHR
SCHEMBL2637908 0.84 NPC1 (0.45) ALDH1A1KMT2AKDM4EMEN1USP2
SCHEMBL2638043 0.83 MAPK10 (0.45) KMT2AMEN1GAAADORA2AADORA2B
SCHEMBL2637445 0.83 NPC1 (0.38) ALDH1A1KMT2AHPGDKDM4EMEN1
SCHEMBL2637520 0.80 DHODH (0.45) KMT2AKDM4EMEN1ALPLALPI
SCHEMBL2637592 0.79 MEN1 (0.45) ALDH1A1KMT2AMEN1SMN1; SMN2NPC1
SCHEMBL2637918 0.79 KMT2A (0.41) ALDH1A1KMT2AKDM4EMEN1MAPK1
SCHEMBL2637500 0.78 ALDH1A1 (0.39) ALDH1A1KMT2AHPGDKDM4EMEN1
SCHEMBL2637350 0.78 ERCC1 (0.48) ALDH1A1KMT2AHPGDKDM4ETSHR
SCHEMBL2637204 0.78 NPC1 (0.43) ALDH1A1KMT2AMEN1MAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2438070-A1 GLYCINE B ANTAGONISTS Merz Pharma GmbH & Co. KGaA (DE) 2012-04-11 EP disclosed
WO-2010139483-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2010-12-09 WO disclosed