SCHEMBL264020

SCHEMBL264020

C=CCn1ccc(=O)n(N)c1=O

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
SLC2A1 P11166 1/20 0.34
ADORA2B P29275 1/20 0.33
KMT2A Q03164 4/20 0.32
NPC1 O15118 4/20 0.32
RAB9A P51151 3/20 0.32
GAA P10253 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CASP3 P42574 1/20 0.32
MEN1 O00255 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GLA P06280 1/20 0.31
HPGD P15428 1/20 0.31
RCE1 Q9Y256 1/20 0.31
CYP19A1 P11511 1/20 0.31
CNR1 P21554 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6028160 0.79 CYP3A4 (0.50) CYP3A4CYP1A2CYP2D6ADORA2BKMT2A
SCHEMBL6675403 0.75 CYP3A4 (0.52) CYP3A4CYP1A2CYP2D6ADORA2BKMT2A
SCHEMBL3807230 0.73 ALDH1A1 (0.41) CYP3A4CYP1A2CYP2D6GAACASP3
SCHEMBL28968571 0.70 CYP3A4 (0.48) CYP3A4CYP1A2CYP2D6ADORA2BKMT2A
SCHEMBL20417809 0.70 SMN1; SMN2 (0.42) CYP3A4CYP1A2CYP2D6SLC2A1KMT2A
SCHEMBL29736630 0.70 KMT2A (0.41) CYP3A4CYP1A2CYP2D6KMT2ANPC1
SCHEMBL7256423 0.68 P2RX4 (0.39) KMT2ANPC1RAB9AGAAMEN1
SCHEMBL1381419 0.67 POLB (0.46) KMT2ANPC1RAB9AGAACASP3
SCHEMBL17563247 0.67 NPC1 (0.40) KMT2ANPC1RAB9AGAASMN1; SMN2
SCHEMBL1567297 0.66 CRBN (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2294076-B1 CHEMICALLY MODIFIED NUCLEOSIDE 5'-TRIPHOSPHATES FOR THERMALLY INITIATED REPLICATION OF NUCLEIC ACID TRILINK BIOTECHNOLOGIES (US) 2017-03-08 EP claimed
EP-2294076-A1 CHEMICALLY MODIFIED NUCLEOSIDE 5'-TRIPHOSPHATES FOR THERMALLY INITIATED AMPLIFICATION OF NUCLEIC ACID TriLink BioTechnologies (US) 2011-03-16 EP claimed
US-20100003724-A1 CHEMICALLY MODIFIED NUCLEOSIDE 5'-TRIPHOSPHATES FOR THERMALLY INITIATED AMPLIFICATION OF NUCLEIC ACID TriLink Bio Technologies 2010-01-07 US claimed
WO-2009151921-A1 CHEMICALLY MODIFIED NUCLEOSIDE 5'-TRIPHOSPHATES FOR THERMALLY INITIATED AMPLIFICATION OF NUCLEIC ACID TRILINK BIOTECHNOLOGIES (US) 2009-12-17 WO claimed
US-20090011488-A1 METHODS FOR STORING COMPOSITIONS USEFUL FOR SYNTHESIZING NUCLEIC ACID MOLECULES ROSETTA INPHARMATICS, LLC (US) 2009-01-08 US claimed
US-20240335551-A1 FUNCTIONAL MOIETIES AND THEIR USES AND SYNTHETIC PREPARATION OLIX US, INC. 2024-10-10 US disclosed
EP-4341269-A1 FUNCTIONAL MOIETIES AND THEIR USES AND SYNTHETIC PREPARATION Olix US, Inc. (US) 2024-03-27 EP disclosed
WO-2022246195-A1 FUNCTIONAL MOIETIES AND THEIR USES AND SYNTHETIC PREPARATION OLIX US, INC. (US) 2022-11-24 WO disclosed
US-20210301324-A1 METHOD FOR ANALYZING FUNCTIONAL SUBUNIT PAIR GENE OF T CELL RECEPTOR AND B CELL RECEPTOR REPERTOIRE GENESIS INCORPORATION (JP) 2021-09-30 US disclosed
EP-3842550-A1 METHOD FOR ANALYZING FUNCTIONAL SUBUNIT PAIR GENE OF T CELL RECEPTOR AND B CELL RECEPTOR Repertoire Genesis Incorporation (JP) 2021-06-30 EP disclosed
US-20190300934-A1 T-CELL RECEPTOR AND B-CELL RECEPTOR REPERTOIRE ANALYSIS SYSTEM USING ONE-STEP REVERSE TRANSCRIPTION TEMPLATE-SWITCHING PCR RIKEN (JP) 2019-10-03 US disclosed
US-20190169679-A1 ONE-STEP REVERSE TRANSCRIPTION TEMPLATE-SWITCHING PCR RIKEN (JP) 2019-06-06 US disclosed
EP-1339699-A1 SUBSTITUTED AMIDOALKYL URACILS AND THE USE THEREOF Bayer Aktiengesellschaft (DE) 2003-09-03 EP disclosed
EP-1303497-A1 SUBSTITUTED AMIDOALKYL-URACILS AS PARP INHIBITORS Bayer Aktiengesellschaft (DE) 2003-04-23 EP disclosed
US-20030022905-A1 Substituted amidoalkyl-uracils and their use BAYER AKTIENGESELLSCHAFT (DE) 2003-01-30 US disclosed
US-20030022905-A1 Substituted amidoalkyl-uracils and their use BAYER AKTIENGESELLSCHAFT (DE) 2003-01-30 US disclosed
WO-2002040455-A8 SUBSTITUTED AMIDOALKYL URACILS AND THEIR USE AS INHIBITORS OF THE POLY(ADP-RIBOSE) SYNTHETASE (PARS) BAYER AG (DE) 2002-07-18 WO disclosed
WO-2002040455-A1 SUBSTITUTED AMIDOALKYL URACILS AND THEIR USE AS INHIBITORS OF THE POLY(ADP-RIBOSE) SYNTHETASE (PARS) BAYER AKTIENGESELLSCHAFT (DE) 2002-05-23 WO disclosed
WO-2002006247-A8 SUBSTITUTED AMIDOALKYL-URACILS AS PARP INHIBITORS BAYER AG (DE) 2002-02-21 WO disclosed
WO-2002006247-A1 SUBSTITUTED AMIDOALKYL-URACILS AS PARP INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2002-01-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240335551-A1 FUNCTIONAL MOIETIES AND THEIR USES AND SYNTHETIC PREPARATION FGB, SELP, PTMS CYP3A4 2842/4885CYP1A2 3659/4885CYP2D6 2428/4885
US-20030022905-A1 Substituted amidoalkyl-uracils and their use UNG, UMPS, TYMP CYP3A4 682/4885CYP1A2 275/4885CYP2D6 114/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.