SCHEMBL26410230

SCHEMBL26410230

COc1ccccc1[C@H]1CCC(=O)O1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.48
HTR2C P28335 3/20 0.45
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
USP2 O75604 1/20 0.44
HTR6 P50406 1/20 0.44
POLL Q9UGP5 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 6/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPT P10636 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
HSD11B1 P28845 1/20 0.43
RECQL P46063 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2B P41595 1/20 0.42
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10569317 1.00 CYP19A1 (0.48) CYP19A1HTR2CMEN1KMT2AUSP2
SCHEMBL28170631 0.80 HCRTR1 (0.43) HTR2CHSD11B1HTR2AHTR2B
SCHEMBL27319090 0.78 CYP19A1 (0.49) CYP19A1HTR2CHTR6ALDH1A1KDM4E
SCHEMBL4310679 0.77 HTR2C (0.49) CYP19A1HTR2CMEN1KMT2AUSP2
SCHEMBL5125493 0.77 HTR2C (0.49) CYP19A1HTR2CMEN1KMT2AUSP2
SCHEMBL13970596 0.76 HTR6 (0.46) CYP19A1HTR2CMEN1KMT2AUSP2
SCHEMBL6414970 0.75 LDHA (0.43) HTR2CHTR6ALDH1A1KDM4ERECQL
SCHEMBL30758308 0.75 ALDH1A1 (0.41) CYP19A1HTR2CMEN1KMT2AHTR6
SCHEMBL16464388 0.74 CYP19A1 (0.50) CYP19A1HTR2CMEN1KMT2AUSP2
SCHEMBL29041073 0.74 HTR2C (0.51) CYP19A1HTR2CMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023192901-A9 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-12-14 WO disclosed
WO-2023192901-A1 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-10-05 WO disclosed