SCHEMBL2641818

SCHEMBL2641818

COc1ccc(/C=C/c2ccnc(F)c2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.61
KDM4E B2RXH2 2/20 0.61
NPC1 O15118 1/20 0.61
CYP3A4 P08684 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2C9 P11712 1/20 0.61
HPGD P15428 1/20 0.61
CYP2C19 P33261 1/20 0.61
RAB9A P51151 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
NFE2L2 Q16236 5/20 0.58
RELA Q04206 5/20 0.57
ESR1 P03372 2/20 0.53
TUBB4A P04350 2/20 0.53
TUBB P07437 2/20 0.53
TUBA3C P0DPH7 2/20 0.53
TUBA1B P68363 2/20 0.53
TUBA4A P68366 2/20 0.53
TUBB4B P68371 2/20 0.53
TUBB3 Q13509 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2641826 1.00 CYP1A2 (0.61) CYP1A2KDM4ENPC1CYP3A4CYP2D6
SCHEMBL29905756 0.83 CYP1A2 (0.65) CYP1A2KDM4ENPC1CYP3A4CYP2D6
SCHEMBL7970832 0.82 LOXL2 (0.45) NPC1HPGDSMN1; SMN2NFE2L2MAPT
SCHEMBL7970830 0.82 LOXL2 (0.45) NPC1HPGDSMN1; SMN2NFE2L2MAPT
SCHEMBL26784184 0.81 CYP1A2 (0.62) CYP1A2KDM4ENPC1CYP3A4CYP2D6
SCHEMBL2879570 0.80 NFE2L2 (0.52) NFE2L2NQO2PTGS2ALOX5PTGS1
SCHEMBL2879571 0.80 NFE2L2 (0.52) NFE2L2NQO2PTGS2ALOX5PTGS1
SCHEMBL13400653 0.80 CYP1A2 (0.61) CYP1A2KDM4ENPC1CYP3A4CYP2D6
SCHEMBL19076282 0.79 HDAC8 (0.49) CYP1A2KDM4ENPC1HPGDRAB9A
SCHEMBL12185880 0.77 NQO2 (0.50) CYP1A2KDM4ENPC1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011141515-A1 DIAGNOSTIC AGENTS FOR AMYLOID BETA IMAGING BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-11-17 WO claimed
WO-2011141515-A1 DIAGNOSTIC AGENTS FOR AMYLOID BETA IMAGING BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-11-17 WO disclosed
WO-2011141515-A1 DIAGNOSTIC AGENTS FOR AMYLOID BETA IMAGING BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-11-17 WO disclosed