SCHEMBL2641819

SCHEMBL2641819

COCOc1ccc(/C=C/c2ccc(F)nc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 2/20 0.51
MAPT P10636 1/20 0.44
KDR P35968 1/20 0.43
RELA Q04206 1/20 0.41
ESR1 P03372 2/20 0.41
AHR P35869 2/20 0.41
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2641825 1.00 NFE2L2 (0.51) NFE2L2MAPTKDRRELAESR1
SCHEMBL2641846 0.85 NFE2L2 (0.67) NFE2L2MAPTRELAESR1AHR
SCHEMBL2641840 0.85 NFE2L2 (0.67) NFE2L2MAPTRELAESR1AHR
SCHEMBL4693722 0.84 RELA (0.53) NFE2L2MAPTRELAESR1AHR
SCHEMBL4693719 0.84 RELA (0.53) NFE2L2MAPTRELAESR1AHR
SCHEMBL12567393 0.84 RELA (0.53) NFE2L2MAPTRELAESR1AHR
SCHEMBL29965553 0.83 CHRNB2 (0.44) NFE2L2
SCHEMBL595487 0.83 CHRNB2 (0.44) NFE2L2
SCHEMBL12567390 0.76 CHRNA7 (0.47) MAPTKDRRELAESR1AHR
SCHEMBL12203894 0.75 ALDH1A1 (0.61) MAPTKDRRELAESR1AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011141515-A1 DIAGNOSTIC AGENTS FOR AMYLOID BETA IMAGING BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-11-17 WO disclosed
WO-2011141515-A1 DIAGNOSTIC AGENTS FOR AMYLOID BETA IMAGING BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-11-17 WO disclosed