SCHEMBL26420142

SCHEMBL26420142

CNC(=O)c1cn(CC(F)(F)F)nc1Cl

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
PDE10A Q9Y233 1/20 0.38
ADORA3 P0DMS8 3/20 0.36
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.34
ADORA2A P29274 2/20 0.34
ADORA1 P30542 2/20 0.34
KLKB1 P03952 9/20 0.34
MAP3K5 Q99683 1/20 0.33
NOTUM Q6P988 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26134353 0.81 ALKBH1 (0.36) LMNAPOLBADORA3ALDH1A1ADORA2A
SCHEMBL26425747 0.81 NPC1 (0.43) LMNAPOLBALDH1A1KDM4E
SCHEMBL7510794 0.77 PDE10A (0.41) LMNAPOLBPDE10AADORA3ALDH1A1
SCHEMBL26134260 0.77 TEAD2 (0.43) ADORA3ALDH1A1KDM4EADORA2AADORA1
SCHEMBL26405871 0.77 CASP1 (0.33) ALDH1A1
SCHEMBL7979529 0.76 GAA (0.46) LMNAPOLBADORA3ALDH1A1ADORA2A
SCHEMBL7510800 0.73 PDE10A (0.42) PDE10AADORA3ALDH1A1KDM4EADORA2A
SCHEMBL26051305 0.71 AR (0.40) PDE10AADORA2AADORA1
SCHEMBL26419959 0.70 KLKB1 (0.43) LMNAPOLBADORA3ALDH1A1KDM4E
SCHEMBL7517096 0.70 L3MBTL1 (0.46) LMNAPOLBPDE10AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023192901-A9 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-12-14 WO disclosed
WO-2023192901-A1 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-10-05 WO disclosed