SCHEMBL264565

SCHEMBL264565

Cc1coc2c(C)ncnc12

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.33
PDGFRB P09619 2/20 0.33
KDR P35968 2/20 0.33
CHRM4 P08173 2/20 0.33
TUBB4A P04350 1/20 0.30
TUBB P07437 1/20 0.30
TUBA3C P0DPH7 1/20 0.30
TUBA1B P68363 1/20 0.30
TUBA4A P68366 1/20 0.30
TUBB4B P68371 1/20 0.30
TUBB3 Q13509 1/20 0.30
TUBB2A Q13885 1/20 0.30
TUBB8 Q3ZCM7 1/20 0.30
TUBA3E Q6PEY2 1/20 0.30
TUBA1A Q71U36 1/20 0.30
TUBA1C Q9BQE3 1/20 0.30
TUBB6 Q9BUF5 1/20 0.30
TUBB2B Q9BVA1 1/20 0.30
TUBB1 Q9H4B7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16576799 0.84 EGFR (0.30) EGFRPDGFRBKDRCHRM4
SCHEMBL2610983 0.79 LIMK1 (0.40) KDR
SCHEMBL12559220 0.75 CHRM4 (0.33) EGFRPDGFRBKDRCHRM4
SCHEMBL16576801 0.69 ELANE (0.33)
SCHEMBL24122008 0.67 CHRM4 (0.36) CHRM4
SCHEMBL12946362 0.67 CYP1A2 (0.36) CHRM4
SCHEMBL2610985 0.65 MEN1 (0.33)
SCHEMBL12559509 0.65 CCR1 (0.38)
SCHEMBL15339503 0.65 IDO1 (0.31)
SCHEMBL8738093 0.65 ELANE (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8163703-B2 Hepatitis C therapies BIOCRYST PHARMACEUTICALS, INC. (US) 2012-04-24 US disclosed
US-8133870-B2 Therapeutic furopyrimidines and thienopyrimidines BIOCRYST PHARMACEUTICALS, INC. (US) 2012-03-13 US disclosed
US-20110144321-A1 SYNTHETIC INTERMEDIATES AND PROCESSES BIOCRYST PHARMACEUTICALS, INC. (US) 2011-06-16 US disclosed
US-20100143300-A1 HEPATITIS C THERAPIES WILMINGTON TRUST, NATIONAL ASSOCIATION 2010-06-10 US disclosed
US-7514410-B2 Hepatitis C therapies BIOCRYST PHARMACEUTICALS, INC. (US) 2009-04-07 US disclosed
US-20080300200-A1 Therapeutic Furopyrimidines and Thienopyrimidines BIOCRYST PHARMACEUTICALS, INC. (US) 2008-12-04 US disclosed
US-7429571-B2 Therapeutic furopyrimidines and thienopyrimidines BIOCRYST PHARMACEUTICALS, INC. (US) 2008-09-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080300200-A1 Therapeutic Furopyrimidines and Thienopyrimidines DPYD, TYMP, TYMS EGFR 970/4885PDGFRB 1290/4885KDR 922/4885
US-20110144321-A1 SYNTHETIC INTERMEDIATES AND PROCESSES G6PD, GALE, UGGT1 EGFR 3358/4885PDGFRB 4283/4885KDR 2548/4885
US-20100143300-A1 HEPATITIS C THERAPIES HAVCR2, FABP1, LIPC EGFR 1952/4885PDGFRB 1535/4885KDR 3621/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.