SCHEMBL26466917

SCHEMBL26466917

Cc1cc(NC(=O)CN2C[C@@H]3C[C@H]2CN3CC(=O)NC(C)(C)C)ccc1F

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.46
TMEM97 Q5BJF2 3/20 0.46
DRD4 P21917 2/20 0.46
CACNA1H O95180 2/20 0.44
DRD3 P35462 2/20 0.41
KCNJ6 P48051 1/20 0.40
KCNJ5 P48544 1/20 0.40
KCNJ3 P48549 1/20 0.40
LTA4H P09960 1/20 0.40
THRB P10828 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26466230 0.88 HTT (0.55) CACNA1HTHRBHPGDTSHRHTT
SCHEMBL26466418 0.88 HTT (0.55) CACNA1HTHRBHPGDTSHRHTT
SCHEMBL26466245 0.88 HTT (0.55) CACNA1HTHRBHPGDTSHRHTT
SCHEMBL26466777 0.86 ALDH1A1 (0.45) CACNA1HLTA4HL3MBTL1TSHRHTT
SCHEMBL26467008 0.85 ALDH1A1 (0.53) CACNA1HL3MBTL1HPGDTSHRHTT
SCHEMBL26466596 0.84 CACNA1H (0.40) SIGMAR1TMEM97DRD4CACNA1HLTA4H
SCHEMBL26466916 0.83 SIGMAR1 (0.42) SIGMAR1TMEM97DRD4CACNA1HDRD3
SCHEMBL26466611 0.82 HTT (0.55) CACNA1HTHRBHPGDTSHRHTT
SCHEMBL26466402 0.81 CACNA1H (0.65) CACNA1H
SCHEMBL26466613 0.81 CACNA1H (0.52) CACNA1HLTA4HL3MBTL1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023192669-A1 T-TYPE CALCIUM CHANNEL MODULATORS COMPRISING A PIPERAZINE OR 1,4-DIAZEPANE CORE AND METHODS OF USE THEREOF PRAXIS PRECISION MEDICINES, INC. (US) 2023-10-05 WO disclosed