SCHEMBL2647337

SCHEMBL2647337

COC(=O)c1cccc2c(C#N)cccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
KDM4E B2RXH2 5/20 0.47
HSD17B10 Q99714 3/20 0.47
IMPDH2 P12268 1/20 0.45
IMPDH1 P20839 1/20 0.45
TSHR P16473 2/20 0.44
LMNA P02545 2/20 0.44
GAA P10253 2/20 0.44
CFTR P13569 1/20 0.43
BRD4 O60885 1/20 0.43
PSMD14 O00487 1/20 0.42
POLB P06746 1/20 0.42
ATM Q13315 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NR4A2 P43354 4/20 0.42
CREBBP Q92793 1/20 0.41
HPGD P15428 2/20 0.41
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5750855 0.90 IMPDH2 (0.53) ALDH1A1KDM4EHSD17B10IMPDH2IMPDH1
SCHEMBL70429 0.84 LMNA (0.59) ALDH1A1KDM4EHSD17B10TSHRLMNA
SCHEMBL181067 0.82 ALDH1A1 (0.55) ALDH1A1KDM4EHSD17B10TSHRLMNA
SCHEMBL2383149 0.81 CA12 (0.48) ALDH1A1KDM4EHSD17B10TSHRLMNA
SCHEMBL30506574 0.81 ALDH1A1 (0.50) ALDH1A1KDM4EHSD17B10TSHRLMNA
SCHEMBL646271 0.81 ALDH1A1 (0.50) ALDH1A1KDM4EHSD17B10TSHRLMNA
SCHEMBL14050225 0.81 ALDH1A1 (0.52) ALDH1A1KDM4EHSD17B10TSHRLMNA
SCHEMBL13209911 0.81 ALDH1A1 (0.47) ALDH1A1KDM4EIMPDH2IMPDH1TSHR
SCHEMBL11281530 0.80 IMPDH2 (0.54) ALDH1A1KDM4EHSD17B10IMPDH2IMPDH1
SCHEMBL1708879 0.80 ALDH1A1 (0.47) ALDH1A1KDM4EHSD17B10TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6613942-B1 Nonpeptide; 4-hydroxy benzoic acid hydrazides NOVO NORDISK A/S (DK) 2003-09-02 US disclosed
EP-1140823-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 2001-10-10 EP disclosed
WO-2000039088-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 2000-07-06 WO disclosed