SCHEMBL2647562

SCHEMBL2647562

O=C(Cc1ccncc1)c1cccc(I)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 1/20 0.48
ALDH1A1 P00352 4/20 0.43
LMNA P02545 2/20 0.43
PLOD2 O00469 3/20 0.42
PLOD3 O60568 3/20 0.42
PLOD1 Q02809 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
CYP2C19 P33261 1/20 0.42
HIF1A Q16665 1/20 0.42
CYP19A1 P11511 1/20 0.41
MAPT P10636 2/20 0.40
GAA P10253 1/20 0.40
VNN1 O95497 1/20 0.39
FNTA P49354 1/20 0.39
FNTB P49356 1/20 0.39
HDAC1 Q13547 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1439664 0.85 MAPT (0.51) ALDH1A1MAPTGAA
SCHEMBL3284705 0.81 KDM4E (0.52) ALDH1A1LMNAMAPTGRM5MEN1
SCHEMBL3073424 0.81 NT5E (0.55) ALDH1A1LMNAHPGDMAPTGAA
SCHEMBL1156959 0.81 CES2 (0.50) ALDH1A1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL1845879 0.81 MAPT (0.49) ALDH1A1LMNAPLOD2PLOD3PLOD1
SCHEMBL6282499 0.79 GRM1 (0.46) ALDH1A1LMNAPLOD2PLOD3PLOD1
SCHEMBL1157353 0.79 ALDH1A1 (0.66) ALDH1A1LMNAPLOD2PLOD3PLOD1
SCHEMBL2477853 0.77 LMNA (0.54) ALDH1A1LMNACYP1A2CYP3A4CYP2D6
SCHEMBL1847397 0.77 GSK3B (0.59) LMNAVNN1GRM5
SCHEMBL2929610 0.77 VNN1 (0.57) ALDH1A1VNN1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0959885-A4 TRIARYL SUBSTITUTED IMIDAZOLES AND METHODS OF USE MERCK & CO INC (US) 2002-07-17 EP disclosed
EP-0959885-A1 TRIARYL SUBSTITUTED IMIDAZOLES AND METHODS OF USE Merck & Co., Inc. (US) 1999-12-01 EP disclosed
WO-1998022108-A1 TRIARYL SUBSTITUTED IMIDAZOLES AND METHODS OF USE MERCK & CO., INC. (US) 1998-05-28 WO disclosed