SCHEMBL2649971

SCHEMBL2649971

O=Cc1cc(Br)c(OCCBr)c(Br)c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
MAPK1 P28482 1/20 0.44
KLK1 P06870 1/20 0.36
THRA P10827 6/20 0.36
THRB P10828 6/20 0.36
ALDH1A3 P47895 2/20 0.35
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
HRH3 Q9Y5N1 2/20 0.34
POLB P06746 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 1/20 0.34
ALDH3A1 P30838 1/20 0.33
FDPS P14324 1/20 0.33
FOXO1 Q12778 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2649949 0.85 ALDH1A1 (0.64) ALDH1A1MAPK1KMT2AMEN1HPGD
SCHEMBL31084168 0.83 ALDH1A1 (0.47) ALDH1A1MAPK1KLK1THRATHRB
SCHEMBL2651217 0.79 SRC (0.47) ALDH1A1MAPK1THRATHRBALDH1A3
SCHEMBL3903040 0.79 THRA (0.57) ALDH1A1MAPK1KLK1THRATHRB
SCHEMBL9858621 0.77 KLK1 (0.41) ALDH1A1KLK1THRATHRBKMT2A
SCHEMBL2650280 0.77 FDPS (0.51) ALDH1A1MAPK1KMT2AMEN1HPGD
SCHEMBL14862481 0.76 HPGD (0.39) ALDH1A1MAPK1KMT2AMEN1HPGD
SCHEMBL7168103 0.76 ALDH1A1 (0.50) ALDH1A1MAPK1THRATHRBKMT2A
SCHEMBL25923588 0.76 MAPT (0.37) ALDH1A1HPGDSMN1; SMN2LMNAMAPT
SCHEMBL13554474 0.76 ALDH1A1 (0.50) ALDH1A1MAPK1THRBALDH1A3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6613942-B1 Nonpeptide; 4-hydroxy benzoic acid hydrazides NOVO NORDISK A/S (DK) 2003-09-02 US disclosed
EP-0994848-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 2000-04-26 EP disclosed
WO-1999001423-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 1999-01-14 WO disclosed
WO-1999001423-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 1999-01-14 WO disclosed