SCHEMBL2650461

SCHEMBL2650461

N#Cc1ccc(F)cc1-c1nc(Cl)ccc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 4/20 0.40
USP8 P40818 1/20 0.39
USP7 Q93009 1/20 0.39
USP47 Q96K76 1/20 0.39
CYP11B1 P15538 2/20 0.38
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
KHK P50053 1/20 0.37
CNR1 P21554 6/20 0.37
KCNQ3 O43525 1/20 0.37
KCNQ2 O43526 1/20 0.37
KCNE1 P15382 1/20 0.37
KCNQ1 P51787 1/20 0.37
CNR2 P34972 3/20 0.37
ALDH1A1 P00352 4/20 0.36
HPGD P15428 4/20 0.36
KDM4E B2RXH2 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2653145 0.88 CNR1 (0.41) CYP11B2USP8USP7USP47GABRA1
SCHEMBL21283227 0.74 MEN1 (0.46) CYP11B2CYP11B1CNR1CNR2ALDH1A1
SCHEMBL21131569 0.74 TRPV4 (0.45) CYP11B2USP8USP7USP47CYP11B1
SCHEMBL9849412 0.73 ADORA1 (0.49) CYP11B2CYP11B1GABRG2GABRB3GABRA5
SCHEMBL6069435 0.70 CNR1 (0.47) CYP11B2CNR1CNR2ALDH1A1HPGD
SCHEMBL31575181 0.69 CYP11B2 (0.41) CYP11B2CYP11B1KHKKCNQ3KCNQ2
SCHEMBL31416799 0.69 CYP11B2 (0.42) CYP11B2CYP11B1KHKKCNQ3KCNQ2
SCHEMBL29311545 0.69 CYP11B2 (0.42) CYP11B2CYP11B1KHKKCNQ3KCNQ2
SCHEMBL24084271 0.69 AR (0.42) CYP11B2USP8USP7USP47CYP11B1
SCHEMBL24084272 0.69 CYP11B2 (0.38) CYP11B2CYP11B1GABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004065388-A1 FLUOROIMIDAZOPYRIMIDINES AS GABA-A ALPHA 2/3 LIGANDS FOR DEPRESSION/ANXIETY MERCK SHARP & DOHME LIMITED (GB) 2004-08-05 WO disclosed