SCHEMBL9849412

SCHEMBL9849412

N#Cc1ccc(Cl)nc1-c1cccc(F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.49
ADORA2A P29274 4/20 0.49
ADORA2B P29275 3/20 0.49
CHUK O15111 1/20 0.48
KDM4E B2RXH2 3/20 0.42
RXFP1 Q9HBX9 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
HPGD P15428 1/20 0.42
MAP4K4 O95819 1/20 0.41
ALDH1A1 P00352 4/20 0.40
HTT P42858 2/20 0.40
LMNA P02545 1/20 0.40
THRB P10828 1/20 0.40
CYP11B2 P19099 3/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
NT5E P21589 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CYP11B1 P15538 1/20 0.39
GABRG2 P18507 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15832010 0.82 ADORA1 (0.49) ADORA1ADORA2AADORA2BCHUKKDM4E
SCHEMBL9849371 0.81 CTSS (0.51) ADORA1ADORA2AKDM4ENPSR1HPGD
SCHEMBL21283227 0.81 MEN1 (0.46) ADORA1ADORA2AADORA2BCHUKKDM4E
SCHEMBL2530034 0.79 ADORA2B (0.47) ADORA1ADORA2AADORA2BCHUKKDM4E
SCHEMBL3290050 0.75 ADORA2B (0.48) ADORA1ADORA2AADORA2BCHUKKDM4E
SCHEMBL11401495 0.74 ADORA1 (0.50) ADORA1ADORA2AADORA2BCHUKKDM4E
SCHEMBL2650461 0.73 CYP11B2 (0.40) KDM4EHPGDALDH1A1CYP11B2CNR1
SCHEMBL1991506 0.71 BCHE (0.46) ADORA1ADORA2AADORA2BCHUKKDM4E
SCHEMBL18357153 0.71 CYP1A2 (0.47) ADORA1ADORA2AADORA2BKDM4ERXFP1
SCHEMBL29907743 0.71 ADORA1 (0.53) ADORA1ADORA2AADORA2BCHUKKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0446604-A2 Pyridine and related aza heterocycle derivatives as cardiovascular agents AMERICAN CYANAMID COMPANY (US) 1991-09-18 EP disclosed