SCHEMBL2650596

SCHEMBL2650596

CC1(C)COB(c2ccc(F)c(-c3ccc(F)cc3)c2)OC1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LPL P06858 1/20 0.43
LIPG Q9Y5X9 1/20 0.43
SNCA P37840 1/20 0.38
MAPK14 Q16539 2/20 0.33
PTGS2 P35354 4/20 0.32
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
PDGFRB P09619 1/20 0.30
KDR P35968 1/20 0.30
PTGS1 P23219 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2649094 0.85 BACE1 (0.37) SNCAMAPK14PTGS1
SCHEMBL1136930 0.81 LPL (0.52) LPLLIPGSNCAPTGS2PTGS1
SCHEMBL20904948 0.81 LIPG (0.68) LPLLIPGPDGFRBKDR
SCHEMBL2658079 0.80 ERN1 (0.42) SNCA
SCHEMBL2649122 0.79 GABRA1 (0.39) SNCA
SCHEMBL2649221 0.79 GABRA1 (0.35) SNCA
SCHEMBL2649142 0.77 PGR (0.38)
SCHEMBL6219095 0.77 SNCA (0.34) SNCA
SCHEMBL5892525 0.76 EGFR (0.39) SNCA
SCHEMBL2659509 0.75 GABRA1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003006464-A1 (1,8) NAPHTHYRIDINES AS GABA LIGANDS, THEIR PHARMACEUTICAL COMPOSITIONS AND USES MERCK SHARP & DOHME LIMITED (GB) 2003-01-23 WO disclosed