SCHEMBL2652007

SCHEMBL2652007

Cc1ccccc1COC([O])c1ccccc1C#N

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.43
MAOB P27338 2/20 0.37
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
LMNA P02545 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
PSMB8 P28062 1/20 0.34
PSMB5 P28074 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2652551 0.88 FFAR1 (0.41) TSHRMAOBKDM4EALDH1A1L3MBTL1
SCHEMBL2652111 0.84 IDO1 (0.41) TSHRMAOBKDM4EALDH1A1
SCHEMBL2652142 0.83 ESR1 (0.42) MAOBKDM4ELMNA
SCHEMBL2652010 0.83 IDO1 (0.40) MAOBL3MBTL1
SCHEMBL2651003 0.83 IDO1 (0.40) MAOBALDH1A1LMNAL3MBTL1
SCHEMBL2650110 0.80 TP53 (0.41) TSHRMAOBKDM4EALDH1A1
SCHEMBL2651078 0.80 IDO1 (0.44) MAOBALDH1A1
SCHEMBL2650879 0.79 ALDH1A1 (0.48) TSHRMAOBALDH1A1LMNA
SCHEMBL2650061 0.77 IDO1 (0.42) TSHRMAOBKDM4EALDH1A1
SCHEMBL2650744 0.76 MAPK14 (0.37) TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1404335-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS Astrazeneca AB (SE) 2004-04-07 EP disclosed
WO-2003000267-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS ASTRAZENECA AB (SE) 2003-01-03 WO disclosed