SCHEMBL2651471

SCHEMBL2651471

[O]C(OCc1cccc(F)c1F)c1cccc(F)c1F

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.38
CES1 P23141 2/20 0.38
FFAR4 Q5NUL3 1/20 0.34
IDO1 P14902 3/20 0.34
ALKBH1 Q13686 1/20 0.34
RIPK1 Q13546 1/20 0.33
OGA O60502 1/20 0.32
ALOX5AP P20292 1/20 0.32
FEN1 P39748 1/20 0.32
AKR1B1 P15121 1/20 0.32
ALDH1A1 P00352 1/20 0.32
BCHE P06276 1/20 0.32
MAOB P27338 2/20 0.31
CXCR2 P25025 1/20 0.31
CCR7 P32248 1/20 0.31
PTGER1 P34995 1/20 0.31
TDO2 P48775 1/20 0.30
DPP4 P27487 1/20 0.30
GLS O94925 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2650998 0.81 CFD (0.39) FFAR4IDO1AKR1B1
SCHEMBL2652478 0.79 IDO1 (0.48) IDO1ALDH1A1MAOBTDO2
SCHEMBL5140181 0.72 IDO1 (0.45) CES2CES1FFAR4IDO1ALKBH1
SCHEMBL2651003 0.71 IDO1 (0.40) IDO1ALDH1A1MAOB
SCHEMBL2642685 0.69 IDO1 (0.42) FFAR4IDO1ALKBH1RIPK1ALDH1A1
SCHEMBL5543468 0.68 IDO1 (0.38) CES2CES1FFAR4IDO1ALKBH1
SCHEMBL323427 0.68 FFAR4 (0.43) CES2CES1FFAR4IDO1ALKBH1
SCHEMBL7193516 0.68 IDO1 (0.38) CES2CES1FFAR4IDO1ALKBH1
SCHEMBL4799320 0.67 RIPK1 (0.34) FFAR4ALKBH1RIPK1OGACXCR2
SCHEMBL2650913 0.67 IDO1 (0.50) FFAR4IDO1ALDH1A1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1404335-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS Astrazeneca AB (SE) 2004-04-07 EP disclosed
WO-2003000267-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS ASTRAZENECA AB (SE) 2003-01-03 WO disclosed