SCHEMBL2651003

SCHEMBL2651003

N#Cc1ccccc1C([O])OCc1ccccc1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.40
ALDH1A1 P00352 3/20 0.37
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KCNH2 Q12809 1/20 0.36
MAPK14 Q16539 1/20 0.35
HTR2A P28223 1/20 0.35
MCL1 Q07820 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
HIF1A Q16665 1/20 0.34
MAOB P27338 3/20 0.34
PARP15 Q460N3 1/20 0.34
PARP14 Q460N5 1/20 0.34
PARP10 Q53GL7 1/20 0.34
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2652551 0.88 FFAR1 (0.41) ALDH1A1TDP1L3MBTL1SMN1; SMN2MAOB
SCHEMBL2650744 0.87 MAPK14 (0.37) ALDH1A1KCNH2MAPK14HTR2APOLB
SCHEMBL2650379 0.86 KAT6A (0.33) IDO1ALDH1A1L3MBTL1HTR2ASMN1; SMN2
SCHEMBL2652111 0.84 IDO1 (0.41) IDO1ALDH1A1SMN1; SMN2MAOBPARP10
SCHEMBL2652478 0.83 IDO1 (0.48) IDO1ALDH1A1MCL1SMN1; SMN2MAOB
SCHEMBL2652010 0.83 IDO1 (0.40) IDO1L3MBTL1MAOBKMT2ANPC1
SCHEMBL2652007 0.83 TSHR (0.43) ALDH1A1L3MBTL1MAOBLMNA
SCHEMBL2651078 0.82 IDO1 (0.44) IDO1ALDH1A1SMN1; SMN2MAOBHTT
SCHEMBL2650713 0.80 MAPK14 (0.37) ALDH1A1KCNH2MAPK14HTR2APOLB
SCHEMBL2650110 0.80 TP53 (0.41) ALDH1A1TDP1MAOBKMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1404335-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS Astrazeneca AB (SE) 2004-04-07 EP disclosed
WO-2003000267-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS ASTRAZENECA AB (SE) 2003-01-03 WO disclosed