SCHEMBL2652478

SCHEMBL2652478

[O]C(OCc1ccccc1F)c1ccccc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.48
ALDH1A1 P00352 2/20 0.44
MAOB P27338 6/20 0.40
PARP15 Q460N3 2/20 0.40
PARP10 Q53GL7 2/20 0.40
PARP14 Q460N5 1/20 0.40
TAAR1 Q96RJ0 1/20 0.38
TDO2 P48775 1/20 0.38
LMNA P02545 3/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MCL1 Q07820 1/20 0.37
MMP1 P03956 1/20 0.37
MMP2 P08253 1/20 0.37
MMP9 P14780 1/20 0.37
MMP12 P39900 1/20 0.37
SLC1A5 Q15758 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2651003 0.83 IDO1 (0.40) IDO1ALDH1A1MAOBPARP15PARP10
SCHEMBL2651471 0.79 CES2 (0.38) IDO1ALDH1A1MAOBTDO2
SCHEMBL10314840 0.73 IDO1 (0.55) IDO1ALDH1A1MAOBPARP15PARP10
SCHEMBL2650913 0.73 IDO1 (0.50) IDO1ALDH1A1PARP10TAAR1TDO2
SCHEMBL2651416 0.72 MMP2 (0.39) IDO1MMP1MMP2MMP9MMP12
SCHEMBL2652142 0.71 ESR1 (0.42) IDO1MAOBTAAR1LMNASLC1A5
SCHEMBL2650236 0.71 IDO1 (0.48) IDO1MAOBTAAR1NPC1RAB9A
SCHEMBL2650544 0.71 IDO1 (0.53) IDO1ALDH1A1MAOBKDM4E
SCHEMBL6204869 0.71 MEN1 (0.41) IDO1ALDH1A1TDO2LMNAMAPT
SCHEMBL2650998 0.70 CFD (0.39) IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1404335-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS Astrazeneca AB (SE) 2004-04-07 EP disclosed
WO-2003000267-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS ASTRAZENECA AB (SE) 2003-01-03 WO disclosed