SCHEMBL26548519

SCHEMBL26548519

COc1ccnc(NC(C)C)c1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.52
CCR5 P51681 1/20 0.52
CCR8 P51685 1/20 0.52
RIOK2 Q9BVS4 7/20 0.49
NOS3 P29474 2/20 0.48
NOS1 P29475 2/20 0.48
NOS2 P35228 2/20 0.48
KDR P35968 1/20 0.47
FDPS P14324 2/20 0.44
PLA2G2A P14555 1/20 0.43
KCNH3 Q9ULD8 1/20 0.42
MAPK10 P53779 4/20 0.42
GSK3A P49840 3/20 0.42
PLAU P00749 1/20 0.41
MAPK14 Q16539 2/20 0.40
HRH4 Q9H3N8 1/20 0.40
TRPV4 Q9HBA0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26550280 0.84 FDPS (0.48) RIOK2KDRFDPSMAPK10MAPK14
SCHEMBL26548744 0.82 NOS1 (0.44) NOS1NOS2FDPSMAPK10MAPK14
SCHEMBL26548751 0.80 MAPK14 (0.40) KDRFDPSMAPK10MAPK14HRH4
Hydrochloric Acid SCHEMBL10980610 0.79 RIOK2 (0.51) CCR1CCR5CCR8RIOK2NOS3
Hydrochloric Acid SCHEMBL10980614 0.79 RIOK2 (0.51) CCR1CCR5CCR8RIOK2NOS3
SCHEMBL3927522 0.79 CCR1 (0.57) CCR1CCR5CCR8RIOK2NOS3
SCHEMBL30496425 0.79 CCR1 (0.57) CCR1CCR5CCR8RIOK2NOS3
SCHEMBL26550285 0.78 MAPK14 (0.41) KDRFDPSMAPK10MAPK14HRH4
SCHEMBL26548746 0.78 FDPS (0.48) FDPSMAPK10MAPK14HRH4
SCHEMBL17700550 0.77 HRH4 (0.50) CCR1CCR5CCR8RIOK2NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023196975-A1 COMPOUNDS THAT INTERACT WITH RAS SUPERFAMILY PROTEINS FOR TREATMENT OF CANCERS, INFLAMMATORY DISEASES, RASOPATHIES, AND FIBROTIC DISEASE SHY THERAPEUTICS, LLC (US) 2023-10-12 WO disclosed