SCHEMBL2655720

SCHEMBL2655720

O=C(C(=O)c1cccc(I)c1)c1ccncc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 1/20 0.56
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
KCNK3 O14649 2/20 0.44
ALDH1A1 P00352 2/20 0.43
PLOD2 O00469 1/20 0.43
PLOD3 O60568 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
PLOD1 Q02809 1/20 0.43
HIF1A Q16665 1/20 0.43
CES2 O00748 5/20 0.42
CES1 P23141 4/20 0.42
NAPRT Q6XQN6 1/20 0.42
GRM5 P41594 1/20 0.42
NT5E P21589 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18079795 0.86 CES2 (0.54) MTORCES2CES1GRM5F2
SCHEMBL15209694 0.84 CES2 (0.61) MTORCES2CES1GRM5HDAC1
SCHEMBL2657896 0.78 MAPT (0.57) MEN1KMT2AKCNK3ALDH1A1PLOD2
SCHEMBL3063840 0.78 NT5E (0.61) MEN1KMT2AKCNK3ALDH1A1HPGD
SCHEMBL3068393 0.78 CES2 (0.74) MEN1KMT2AALDH1A1CYP1A2CYP3A4
SCHEMBL3074392 0.78 KMT2A (0.74) MEN1KMT2AKCNK3ALDH1A1PLOD2
SCHEMBL2783342 0.77 NAPRT (0.65) MEN1KMT2AALDH1A1PLOD2PLOD3
SCHEMBL29875488 0.76 MTOR (0.44) MTORCES2CES1GRM5F2
SCHEMBL2647562 0.76 MTOR (0.48) MTORMEN1KMT2AALDH1A1PLOD2
SCHEMBL30967896 0.75 MGLL (0.42) MTORCES2CES1GRM5F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0959885-A4 TRIARYL SUBSTITUTED IMIDAZOLES AND METHODS OF USE MERCK & CO INC (US) 2002-07-17 EP disclosed
EP-0959885-A1 TRIARYL SUBSTITUTED IMIDAZOLES AND METHODS OF USE Merck & Co., Inc. (US) 1999-12-01 EP disclosed
WO-1998022108-A1 TRIARYL SUBSTITUTED IMIDAZOLES AND METHODS OF USE MERCK & CO., INC. (US) 1998-05-28 WO disclosed