SCHEMBL2656867

SCHEMBL2656867

NC(=O)CCCCCc1nccs1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.46
PLA2G4A P47712 3/20 0.43
FDPS P14324 1/20 0.40
ALDH1A1 P00352 2/20 0.36
TSHR P16473 2/20 0.36
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TBXAS1 P24557 3/20 0.35
PKM P14618 1/20 0.35
HSD17B10 Q99714 1/20 0.35
COPS5 Q92905 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2657137 0.98 PLA2G4A (0.44) CES1PLA2G4AFDPSALDH1A1TSHR
SCHEMBL175216 0.87 FDPS (0.43) CES1PLA2G4AFDPSALDH1A1TSHR
SCHEMBL7174088 0.86 CES1 (0.49) CES1PLA2G4ATBXAS1
Hydrochloric Acid SCHEMBL31146299 0.86 FDPS (0.42) CES1PLA2G4AFDPSALDH1A1TSHR
SCHEMBL11156307 0.84 PLA2G4A (0.48) CES1PLA2G4ATBXAS1
SCHEMBL19929602 0.83 PLA2G4A (0.43) CES1PLA2G4AFDPSALDH1A1TSHR
Urea SCHEMBL7180010 0.81 PLA2G4A (0.45) PLA2G4AFDPSALDH1A1POLBSMN1; SMN2
SCHEMBL7184826 0.81 COPS5 (0.39) CES1FDPSALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL6179956 0.79 SMN1; SMN2 (0.44) CES1PLA2G4AFDPSALDH1A1SMN1; SMN2
SCHEMBL7275156 0.78 FDPS (0.41) CES1PLA2G4AFDPSALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2091947-A2 GLUCOKINASE ACTIVATORS Takeda San Diego, Inc. (US) 2009-08-26 EP claimed
WO-2008079787-A2 GLUCOKINASE ACTIVATORS TAKEDA SAN DIEGO, INC. (US) 2008-07-03 WO claimed
EP-2091947-A2 GLUCOKINASE ACTIVATORS Takeda San Diego, Inc. (US) 2009-08-26 EP disclosed
WO-2008079787-A2 GLUCOKINASE ACTIVATORS TAKEDA SAN DIEGO, INC. (US) 2008-07-03 WO disclosed