SCHEMBL2659614

SCHEMBL2659614

Cc1ccsc1S(=O)(=O)Nc1cccc2cc(C(=O)NCC3(O)CCN(Cc4ccccc4)CC3)[nH]c12

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.37
LMNA P02545 2/20 0.37
TP53 P04637 2/20 0.37
NPFFR1 Q9GZQ6 4/20 0.37
NPFFR2 Q9Y5X5 4/20 0.37
ACHE P22303 3/20 0.35
MAOB P27338 2/20 0.35
PKM P14618 1/20 0.35
ALOX5 P09917 1/20 0.35
BACE1 P56817 1/20 0.35
UTS2R Q9UKP6 1/20 0.35
THRB P10828 1/20 0.35
MAOA P21397 1/20 0.35
RAB9A P51151 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRK1 P41145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2659433 0.82 NSD2 (0.33) NAMPTLMNATP53THRB
SCHEMBL2661008 0.80 NSD2 (0.33)
SCHEMBL2660248 0.80 NSD2 (0.33) RAB9A
SCHEMBL2659954 0.79 NSD2 (0.32)
SCHEMBL2661515 0.78 MAPK8 (0.33) LMNATP53RAB9A
SCHEMBL2659616 0.77 CCR5 (0.40) NAMPTLMNATP53NPFFR1NPFFR2
SCHEMBL2660564 0.76 KDM4E (0.37) LMNARAB9A
SCHEMBL2659423 0.76 HRH4 (0.32) LMNATP53PKMTHRB
SCHEMBL2659185 0.76 HPGD (0.40)
SCHEMBL2659015 0.76 HDAC3 (0.32) LMNATP53PKMTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074119-A1 INDOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008050821-A1 INDOLE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-02 WO disclosed