SCHEMBL2659634

SCHEMBL2659634

COCCOc1cc(NS(=O)(=O)c2ncccc2C)c2[nH]c(C(=O)NCC3(SCc4ccccc4)CCOCC3)cc2c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.34
LMNA P02545 3/20 0.34
TP53 P04637 2/20 0.34
THRB P10828 2/20 0.34
ALDH1A1 P00352 1/20 0.32
RAB9A P51151 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ITGB3 P05106 3/20 0.32
ITGA2B P08514 3/20 0.32
ITGAV P06756 1/20 0.32
SYK P43405 1/20 0.31
KDM4E B2RXH2 2/20 0.31
SLC40A1 Q9NP59 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2660662 0.92 MAPT (0.34) MAPTLMNATP53THRBRAB9A
SCHEMBL2660175 0.81 MAPT (0.35) MAPTLMNATP53THRBALDH1A1
SCHEMBL2661032 0.81 MAPT (0.35) MAPTLMNATP53THRBRAB9A
SCHEMBL2660116 0.81 MAPT (0.41) MAPTLMNATP53THRBSLC40A1
SCHEMBL2659522 0.81 SLC40A1 (0.38) MAPTLMNATP53THRBALDH1A1
SCHEMBL2659636 0.81 MAPT (0.34) MAPTLMNATP53THRBALDH1A1
SCHEMBL2660335 0.80 MAPT (0.34) MAPTLMNATP53THRBRAB9A
SCHEMBL2659586 0.79 MAPT (0.36) MAPTLMNATP53THRBALDH1A1
SCHEMBL2659404 0.78 LMNA (0.33) MAPTLMNATP53THRBITGB3
SCHEMBL2659714 0.77 SLC40A1 (0.38) MAPTLMNATP53THRBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074119-A1 INDOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008050821-A1 INDOLE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-02 WO disclosed