SCHEMBL2660958

SCHEMBL2660958

COC(=O)C(Cc1nccn1C)Nc1ccccc1N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.43
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
TP53 P04637 2/20 0.37
LDHA P00338 1/20 0.37
LDHB P07195 1/20 0.37
CYP26A1 O43174 1/20 0.36
HDAC2 Q92769 4/20 0.36
HDAC6 Q9UBN7 3/20 0.36
HDAC3 O15379 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC4 P56524 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
THRB P10828 1/20 0.35
ITGB1 P05556 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2516349 0.82 KMT2A (0.42) KMT2ACYP26A1HPGD
SCHEMBL25647654 0.74 FDPS (0.40) KMT2AMEN1LDHALDHBSMN1; SMN2
Hydrochloric Acid SCHEMBL25222775 0.73 FDPS (0.39) KMT2AMEN1LDHALDHBSMN1; SMN2
SCHEMBL25227617 0.70 KLK5 (0.43) ITGA4ITGB7
SCHEMBL31146320 0.68 PSMB5 (0.47) HDAC1HDAC2HDAC6HDAC3HDAC8
SCHEMBL25225956 0.68 PSMB5 (0.47) HDAC1HDAC2HDAC6HDAC3HDAC8
SCHEMBL27980070 0.67 FDPS (0.41) KMT2AMEN1TP53LDHALDHB
SCHEMBL18117397 0.67 FDPS (0.38) KMT2AMEN1LDHALDHBSMN1; SMN2
SCHEMBL14853086 0.67 FDPS (0.38) KMT2AMEN1LDHALDHBSMN1; SMN2
SCHEMBL690630 0.67 ITGA4 (0.43) KMT2AMEN1LDHALDHBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001875-A2 GLUCOKINASE ACTIVATORS Takeda San Diego, Inc. (US) 2008-12-17 EP disclosed
WO-2007104034-A2 GLUCOKINASE ACTIVATORS TAKEDA SAN DIEGO, INC. (US) 2007-09-13 WO disclosed