SCHEMBL26645835

SCHEMBL26645835

Fc1c(-c2c[c]ccn2)ccc2ccccc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.37
MAPK14 Q16539 3/20 0.37
CSNK1D P48730 2/20 0.37
CSNK1E P49674 2/20 0.37
CYP3A4 P08684 3/20 0.35
ALDH1A1 P00352 3/20 0.33
MAPT P10636 3/20 0.33
HSD17B10 Q99714 2/20 0.33
KDM4E B2RXH2 2/20 0.33
NPC1 O15118 2/20 0.33
TP53 P04637 2/20 0.33
HPGD P15428 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
CYP2A6 P11509 2/20 0.33
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
RAB9A P51151 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
MAPK1 P28482 2/20 0.33
CYP17A1 P05093 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28108385 0.80 KDM4E (0.45) ALDH1A1MAPTHSD17B10KDM4ENPC1
SCHEMBL31589324 0.75 ALDH1A1 (0.58) HSD11B1MAPK14CSNK1DCSNK1ECYP3A4
SCHEMBL2751007 0.73 CDK2 (0.38) HSD11B1NPC1MAPK1GSK3BCDK5
SCHEMBL28725076 0.70 HTR2C (0.35) ALDH1A1MAPTHSD17B10KDM4ENPC1
SCHEMBL5780140 0.69 IDO1 (0.43) HSD11B1MAPK14CYP3A4ALDH1A1NPC1
SCHEMBL8100099 0.69 TGFBR1 (0.46) MAPK14CSNK1DALDH1A1MAPTHSD17B10
SCHEMBL2753034 0.69 KMO (0.44) NPC1TP53RAB9A
SCHEMBL27779509 0.68 ALDH1A1 (0.48) HSD11B1MAPK14CSNK1DCSNK1ECYP3A4
SCHEMBL2752979 0.67 GABRA1 (0.33) KDM4ENPC1TP53SMN1; SMN2TDP1
SCHEMBL4006504 0.67 CYP1A2 (0.47) ALDH1A1MAPTHSD17B10KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023213882-A1 IRREVERSIBLE MUTEGFR INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2023-11-09 WO disclosed