SCHEMBL266510

SCHEMBL266510

O=C1CCc2cc(O)ccc2C1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.54
DRD1 P21728 11/20 0.53
DRD2 P14416 10/20 0.53
DRD5 P21918 9/20 0.53
DRD3 P35462 8/20 0.53
PBRM1 Q86U86 1/20 0.52
DRD4 P21917 6/20 0.47
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP11B1 P15538 2/20 0.46
CYP11B2 P19099 2/20 0.46
CYP2C19 P33261 2/20 0.46
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
PRKCI P41743 1/20 0.44
OPRK1 P41145 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30199197 0.92 CYP2A6 (0.54) CYP2A6DRD1DRD2DRD5DRD3
SCHEMBL266616 0.92 CYP2A6 (0.54) CYP2A6DRD1DRD2DRD5DRD3
SCHEMBL13590991 0.85 CYP1A2 (0.50) DRD1DRD2DRD5DRD3PBRM1
SCHEMBL8408108 0.79
SCHEMBL588130 0.79 CYP2A6 (0.54) CYP2A6CYP1A2CYP3A4CYP2C9CYP11B1
Ammonia Solution, Strong SCHEMBL21632258 0.77 DRD2 (0.54) DRD1DRD2DRD5DRD3PBRM1
SCHEMBL6903685 0.77 DRD1 (0.76) CYP2A6DRD1DRD2DRD5DRD3
SCHEMBL1701852 0.75 CYP2A6 (0.54) CYP2A6CYP1A2CYP3A4CYP2C9CYP11B1
SCHEMBL12152856 0.75 CYP2A6 (0.54) CYP2A6PBRM1CYP1A2CYP3A4CYP2C9
SCHEMBL354022 0.75 CYP2A6 (0.54) CYP2A6CYP1A2CYP3A4CYP2C9CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 54 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117586289-A Preparation method of 2- (6- (benzyloxy) -3, 4-dihydronaphthalene-2-yl) -4, 5-5-tetramethyl-1, 3, 2-dioxaborane 四川新迪生物制药有限公司 2024-02-23 CN claimed
CN-116969848-A Preparation method of intermediate of drug for treating advanced breast cancer 北京康立生医药技术开发有限公司 2023-10-31 CN claimed
CN-122059824-A Synthesis method of ilalastyl chiral intermediate 上海格苓凯生物科技有限公司 2026-05-19 CN disclosed
US-20260035339-A1 TETRAHYDRONAPHTHALENE DERIVATIVE ATRANSEN PHARMA LTD (JP) 2026-02-05 US disclosed
CN-116969848-B Preparation method of intermediate of drug for treating advanced breast cancer 北京康立生医药技术开发有限公司 2025-12-12 CN disclosed
CN-119569588-A Preparation method and intermediate of ilast hydrochloride 杭州诺澳生物医药科技有限公司 2025-03-07 CN disclosed
EP-4501906-A1 TETRAHYDRONAPHTHALENE DERIVATIVE Atransen Pharma Ltd. (JP) 2025-02-05 EP disclosed
CN-119100936-A In the ilast group Synthesis method of intermediate 杭州诺澳生物医药科技有限公司 2024-12-10 CN disclosed
CN-118974007-A Tetrahydronaphthalene derivatives 阿创森制药股份有限公司 2024-11-15 CN disclosed
CN-118702588-A Preparation method of ilast and intermediate thereof 重庆华邦胜凯制药有限公司 2024-09-27 CN disclosed
WO-2024175615-A1 DIHYDRONAPTHALENE DERIVATIVES MERCK PATENT GMBH (DE) 2024-08-29 WO disclosed
CN-1756746-A 6-substituted nicotinamide derivatives as opioid receptor antagonists LILLY CO ELI (US) 2006-04-05 CN disclosed
EP-1613597-A1 6-SUBSTITUTED NICOTINAMIDE DERIVATIVES AS OPIOID RECEPTOR ANTAGONISTS Eli Lilly and Company (US) 2006-01-11 EP disclosed
EP-1569645-A2 METHOD OF USING AMINOCYANOPYRIDINE COMPOUNDS AS MITOGEN ACTIVATED PROTEIN KINASE-ACTIVATED PROTEIN KINASE-2 INHIBITORS Pharmacia Corporation (US) 2005-09-07 EP disclosed
EP-1569932-A1 AMINOCYANOPYRIDINE INHIBITORS OF MITOGEN ACTIVATED PROTEIN KINASE-ACTIVATED PROTEIN KINASE-2 Pharmacia Corporation (US) 2005-09-07 EP disclosed
WO-2004080968-A1 6-SUBSTITUTED NICOTINAMIDE DERIVATIVES AS OPIOID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2004-09-23 WO disclosed
US-20040142978-A1 Aminocyanopyridine inhibitors of mitogen activated protein kinase-activated protein kinase-2 PHARMACIA CORPORATION (US) 2004-07-22 US disclosed
WO-2004055015-A1 AMINOCYANOPYRIDINE INHIBITORS OF MITOGEN ACTIVATED PROTEIN KINASE-ACTIVATED PROTEIN KINASE-2 PHARMACIA CORPORATION (US) 2004-07-01 WO disclosed
WO-2004054505-A2 METHOD OF USING AMINOCYANOPYRIDINE COMPOUNDS AS MITOGEN ACTIVATED PROTEIN KINASE-ACTIVATED PROTEIN KINASE-2 INHIBITORS PHARMACIA CORPORATION (US) 2004-07-01 WO disclosed
US-20040127519-A1 Method of using aminocyanopyridine compounds as mitogen activated protein kinase-activated protein kinase-2 inhibitors PHARMACIA CORPORATION 2004-07-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040127519-A1 Method of using aminocyanopyridine compounds as mitogen activated protein kinase-activated protein kinase-2 inhibitors MAPKAPK2, MAP2K2, MAP3K2 CYP2A6 2913/4885DRD1 4132/4885DRD2 3188/4885
US-20040142978-A1 Aminocyanopyridine inhibitors of mitogen activated protein kinase-activated protein kinase-2 MAP4K2, MAP3K20, MAPKAPK2 CYP2A6 3903/4885DRD1 4330/4885DRD2 3273/4885
US-20260035339-A1 TETRAHYDRONAPHTHALENE DERIVATIVE LATS1, LATS2, BCAT1 CYP2A6 1376/4885DRD1 3554/4885DRD2 4449/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.