SCHEMBL2666271

SCHEMBL2666271

Cc1ccnc(-c2cc(F)ccc2F)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.41
CYP3A4 P08684 3/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C19 P33261 2/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
MEN1 O00255 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
NPC1 O15118 1/20 0.37
POLB P06746 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TGFBR1 P36897 4/20 0.36
FFAR1 O14842 1/20 0.36
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
CYP2C8 P10632 1/20 0.36
NPY5R Q15761 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8365562 0.85 TGFBR1 (0.41) CYP3A4CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL2666247 0.81 FFAR1 (0.40) CYP3A4CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL2666288 0.81 CYP1A2 (0.49) CYP3A4CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL8365573 0.80 HSD11B1 (0.43) CYP3A4CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL8365560 0.80 GRM5 (0.41) CYP3A4CYP1A2ALDH1A1FFAR1
SCHEMBL8363964 0.79 CYP1A2 (0.44) CYP3A4CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL31517722 0.77 CASP6 (0.43) IDH1KMT2AL3MBTL1TGFBR1NPY5R
SCHEMBL8365589 0.77 FFAR1 (0.36) CYP3A4CYP1A2CYP2D6CYP2C19ALDH1A1
SCHEMBL2666248 0.77 KMO (0.47) KMT2AL3MBTL1MEN1NPC1RAB9A
SCHEMBL8363956 0.74 KMT2A (0.56) CYP3A4CYP1A2CYP2D6CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002076983-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 2002-10-03 WO disclosed