SCHEMBL26684635

SCHEMBL26684635

NC(=O)c1nc(Cl)cc(C(F)(F)F)c1N

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
JUN P05412 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
LIMK1 P53667 4/20 0.37
CFTR P13569 5/20 0.36
IKBKB O14920 3/20 0.36
LMNA P02545 1/20 0.35
SCN9A Q15858 1/20 0.34
MBOAT4 Q96T53 1/20 0.34
JAK2 O60674 1/20 0.33
CASP1 P29466 1/20 0.33
CHEK2 O96017 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26852629 0.80 HPGD (0.43) LIMK1CFTRIKBKBLMNAMBOAT4
SCHEMBL30516416 0.77 LMNA (0.41) IKBKBLMNA
SCHEMBL565623 0.75 POLB (0.46) JUNNFKB1NFKB2RELALIMK1
SCHEMBL13076777 0.74 PIK3CD (0.41)
SCHEMBL31028563 0.74 PIK3CD (0.41)
SCHEMBL18109672 0.74 POLB (0.44) LIMK1IKBKBLMNA
SCHEMBL30609423 0.74 LMNA (0.38) LIMK1IKBKBLMNA
SCHEMBL24558660 0.71 LMNA (0.36) IKBKBLMNAJAK2
SCHEMBL30397207 0.71 ALDH1A1 (0.39) CFTRIKBKBLMNASCN9ACASP1
SCHEMBL29028859 0.71 ALDH1A1 (0.39) CFTRIKBKBLMNASCN9ACASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250282785-A1 PYRROLIDINONE DERIVATIVES AS INHIBITORS OF NF KAPPA B INDUCING KINASE JANSSEN PHARMACEUTICA NV (BE) 2025-09-11 US disclosed
EP-4522608-A1 PYRROLIDINONE DERIVATIVES AS INHIBITORS OF NF KAPPA B INDUCING KINASE JANSSEN Pharmaceutica NV (BE) 2025-03-19 EP disclosed
CN-119546602-A Pyrrolidone derivatives as inhibitors of nfkb-induced kinase 詹森药业有限公司 2025-02-28 CN disclosed
WO-2023217906-A1 PYRROLIDINONE DERIVATIVES AS INHIBITORS OF NF KAPPA B INDUCING KINASE JANSSEN PHARMACEUTICA NV (BE) 2023-11-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250282785-A1 PYRROLIDINONE DERIVATIVES AS INHIBITORS OF NF KAPPA B INDUCING KINASE NFKBIA, IKBKG, IKBKB JUN 713/4885NFKB1 4/4885NFKB2 8/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.