SCHEMBL26697254

SCHEMBL26697254

O=C(Nc1ccncc1)Nc1ccc(O)cc1Cl

nearest known ligand 0.76

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 9/20 0.72
POLB P06746 1/20 0.66
MEN1 O00255 8/20 0.62
MDM2 Q00987 1/20 0.58
SMARCA2 P51531 1/20 0.55
SMARCA4 P51532 1/20 0.55
MAPT P10636 3/20 0.55
HTT P42858 3/20 0.55
LMNA P02545 1/20 0.55
GRIK1 P39086 1/20 0.55
TAAR1 Q96RJ0 2/20 0.51
KDM4E B2RXH2 1/20 0.51
MAPK1 P28482 1/20 0.51
ALDH1A1 P00352 1/20 0.50
KDR P35968 1/20 0.48
BCHE P06276 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5640255 0.86 KMT2A (0.78) KMT2APOLBMEN1MDM2SMARCA2
SCHEMBL21750979 0.84 MAOA (0.61) KMT2APOLBMEN1MAPTHTT
SCHEMBL29757943 0.84 MAOA (0.61) KMT2APOLBMEN1MAPTHTT
SCHEMBL26697246 0.82 KMT2A (0.56) KMT2APOLBMEN1MAPTHTT
SCHEMBL21750906 0.82 RAB9A (0.56) KMT2APOLBMEN1HTTGRIK1
SCHEMBL29757932 0.82 RAB9A (0.56) KMT2APOLBMEN1HTTGRIK1
SCHEMBL26697260 0.81 CA12 (0.64) KMT2AMEN1MAPTHTTGRIK1
SCHEMBL26697200 0.79 GRIK1 (0.58) KMT2APOLBMEN1MAPTLMNA
SCHEMBL14514332 0.79 KMT2A (0.64) KMT2APOLBMEN1MAPTHTT
SCHEMBL195117 0.76 KMT2A (0.67) KMT2APOLBMEN1MDM2SMARCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114920703-B Quinazoline derivative and preparation method and application thereof 天津济坤医药科技有限公司 2024-01-09 CN disclosed
WO-2023226323-A1 QUINAZOLINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 天津济坤医药科技有限公司 2023-11-30 WO disclosed
WO-2023226323-A1 QUINAZOLINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 天津济坤医药科技有限公司 2023-11-30 WO disclosed
CN-114920703-A Quinazoline derivative and preparation method and application thereof 天津济坤医药科技有限公司 2022-08-19 CN disclosed