SCHEMBL26697246

SCHEMBL26697246

Cc1ccc(NC(=O)Nc2ccc(O)cc2Cl)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.56
RAB9A P51151 5/20 0.56
MEN1 O00255 5/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
NPC1 O15118 3/20 0.56
LMNA P02545 2/20 0.56
HTT P42858 2/20 0.56
ALDH1A1 P00352 3/20 0.56
MAPT P10636 2/20 0.56
CXCR2 P25025 2/20 0.52
TRPV1 Q8NER1 4/20 0.51
GAA P10253 2/20 0.50
ALOX12 P18054 1/20 0.50
KDM4E B2RXH2 1/20 0.49
HPGD P15428 1/20 0.49
GRIK1 P39086 1/20 0.49
PDK1 Q15118 1/20 0.49
PDK2 Q15119 1/20 0.49
PDK3 Q15120 1/20 0.49
PDK4 Q16654 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29757932 0.85 RAB9A (0.56) KMT2ARAB9AMEN1SMN1; SMN2NPC1
SCHEMBL21750906 0.85 RAB9A (0.56) KMT2ARAB9AMEN1SMN1; SMN2NPC1
SCHEMBL21750979 0.84 MAOA (0.61) KMT2ARAB9AMEN1SMN1; SMN2NPC1
SCHEMBL29757943 0.84 MAOA (0.61) KMT2ARAB9AMEN1SMN1; SMN2NPC1
SCHEMBL26697200 0.82 GRIK1 (0.58) KMT2ARAB9AMEN1SMN1; SMN2NPC1
SCHEMBL26697279 0.82 NPC1 (0.53) KMT2ARAB9AMEN1SMN1; SMN2NPC1
SCHEMBL26697254 0.82 KMT2A (0.72) KMT2AMEN1LMNAHTTALDH1A1
SCHEMBL26697260 0.81 CA12 (0.64) KMT2ARAB9AMEN1HTTMAPT
SCHEMBL26697245 0.81 RAB9A (0.53) KMT2ARAB9AMEN1SMN1; SMN2NPC1
SCHEMBL1310905 0.80 MAOA (0.67) KMT2ARAB9AMEN1SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114920703-B Quinazoline derivative and preparation method and application thereof 天津济坤医药科技有限公司 2024-01-09 CN disclosed
WO-2023226323-A1 QUINAZOLINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 天津济坤医药科技有限公司 2023-11-30 WO disclosed
WO-2023226323-A1 QUINAZOLINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USE THEREOF 天津济坤医药科技有限公司 2023-11-30 WO disclosed
CN-114920703-A Quinazoline derivative and preparation method and application thereof 天津济坤医药科技有限公司 2022-08-19 CN disclosed