SCHEMBL2669899

SCHEMBL2669899

CCCCCC(C)C(Nc1ccc(C(=O)N(C)CCC(=O)O)cc1)c1oc2ccc(F)cc2c1COCCOC

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.36
CCKAR P32238 1/20 0.32
GCG P01275 1/20 0.31
ABCB11 O95342 1/20 0.31
CYP3A4 P08684 1/20 0.31
ADRA2B P18089 1/20 0.31
OPRD1 P41143 1/20 0.31
SCN5A Q14524 1/20 0.31
PTGDR2 Q9Y5Y4 2/20 0.31
P2RY12 Q9H244 2/20 0.31
LTB4R Q15722 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
PIK3CD O00329 1/20 0.30
PIK3CA P42336 1/20 0.30
PIK3CB P42338 1/20 0.30
PIK3CG P48736 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2669847 0.87 NAMPT (0.36) NAMPTGCGHDAC6PIK3CBHDAC3
SCHEMBL2669769 0.86 NAMPT (0.36) NAMPTGCGPTGDR2HDAC6PIK3CB
SCHEMBL2669810 0.85 NAMPT (0.34) NAMPTPIK3CB
SCHEMBL2669784 0.82 NAMPT (0.33) NAMPTABCB11CYP3A4ADRA2BOPRD1
SCHEMBL13069831 0.82 NPC1 (0.33) CCKARLTB4R
SCHEMBL2669939 0.82 NPC1 (0.39) ABCB11
SCHEMBL3402059 0.80 NAMPT (0.38) NAMPTGCGPIK3CDPIK3CAPIK3CB
SCHEMBL2669959 0.80 SRC (0.33) NAMPTCCKARP2RY12
SCHEMBL2669941 0.78 TP53 (0.36) NAMPTPIK3CBHDAC3HDAC1
SCHEMBL723029 0.77 NAMPT (0.35) NAMPTPTGDR2PIK3CDPIK3CAPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009110520-A1 HETEROCYCLIC COMPOUND 武田薬品工業株式会社 (JP) 2009-09-11 WO disclosed