SCHEMBL26918921

SCHEMBL26918921

O=C(O)N1CCC(Nc2ncc(C(F)(F)F)c(OC3CCOC3)n2)CC1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 3/20 0.42
MAPK3 P27361 3/20 0.41
MAPK1 P28482 1/20 0.41
CDK1 P06493 1/20 0.41
CCNB1 P14635 1/20 0.41
CCNE1 P24864 1/20 0.41
CDK2 P24941 1/20 0.41
LRRK2 Q5S007 4/20 0.40
ULK1 O75385 1/20 0.40
CCNK O75909 1/20 0.40
CDK12 Q9NYV4 1/20 0.40
EGFR P00533 3/20 0.39
EPHX2 P34913 2/20 0.39
HSD11B1 P28845 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26918911 1.00 PTK2 (0.42) PTK2MAPK3MAPK1CDK1CCNB1
SCHEMBL30697139 0.88 IDH1 (0.44) PTK2MAPK3MAPK1CDK1CCNB1
SCHEMBL26919164 0.86 AXL (0.43) CDK1CCNB1CCNE1CDK2LRRK2
SCHEMBL26919173 0.86 AXL (0.43) CDK1CCNB1CCNE1CDK2LRRK2
SCHEMBL29763036 0.86 AXL (0.43) CDK1CCNB1CCNE1CDK2LRRK2
SCHEMBL26920123 0.82 ULK1 (0.44) PTK2MAPK3MAPK1CDK1CCNB1
SCHEMBL26920117 0.82 ULK1 (0.44) PTK2MAPK3MAPK1CDK1CCNB1
SCHEMBL29763071 0.82 ULK1 (0.44) PTK2MAPK3MAPK1CDK1CCNB1
SCHEMBL29763020 0.81 CCR6 (0.42) MAPK1CDK1CCNB1CCNE1CDK2
SCHEMBL22998319 0.79 ULK1 (0.44) PTK2MAPK3MAPK1CDK1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4289835-A1 CDK INHIBITOR Shanghai Qilu Pharmaceutical Research and Development Centre Ltd. (CN) 2023-12-13 EP disclosed
CN-116472270-A CDK inhibitors 上海齐鲁制药研究中心有限公司 2023-07-21 CN disclosed